SCHEMBL24769737

SCHEMBL24769737

c1csc(Cc2cncnc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.51
PLA2G7 Q13093 3/20 0.44
TAAR1 Q96RJ0 1/20 0.41
TSHR P16473 3/20 0.40
LMNA P02545 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
CYP1A2 P05177 4/20 0.38
CYP3A4 P08684 4/20 0.38
CYP2D6 P10635 4/20 0.38
ALDH1A1 P00352 4/20 0.38
CYP2C19 P33261 3/20 0.38
CYP2C9 P11712 3/20 0.38
MAPK1 P28482 2/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306418 0.81 ADRA1D (0.49) ADRA1DLMNACYP1A2CYP3A4CYP2D6
SCHEMBL6645686 0.79 CYP17A1 (0.56) ADRA1DTAAR1TSHRLMNAADRA2A
SCHEMBL25185325 0.77 ADRA1D (0.45) ADRA1DTAAR1TSHRLMNACYP1A2
SCHEMBL559559 0.75 TAAR1 (0.56) ADRA1DTAAR1TSHRLMNAADRA2A
SCHEMBL28301068 0.74 EGFR (0.44) ADRA1DTSHRLMNACYP1A2CYP3A4
SCHEMBL45228 0.74 LMNA (0.50) ADRA1DTAAR1TSHRLMNAALDH1A1
Ammonia Solution, Strong SCHEMBL27757668 0.72 LMNA (0.49) ADRA1DTAAR1TSHRLMNAALDH1A1
Methane SCHEMBL11161392 0.72 LMNA (0.49) ADRA1DTAAR1TSHRLMNAALDH1A1
SCHEMBL9825918 0.72 LMNA (0.49) ADRA1DTAAR1TSHRLMNAALDH1A1
SCHEMBL28205872 0.72 ADRA1D (0.47) ADRA1DTAAR1TSHRLMNAADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022263800-A1 PROCESS JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2022-12-22 WO disclosed
CN-101918358-B Novel vitamin D receptor activators and methods of manufacture ABBVIE (US) 2015-10-14 CN disclosed
CN-104211626-A NEW VITAMIN D RECEPTOR ACTIVATORS AND METHODS OF MAKING ABBVIE INC 2014-12-17 CN disclosed
CN-102816165-A Amino-aza-adamantane derivatives and methods of use ABBOTT LAB 2012-12-12 CN disclosed
CN-101925599-A Azabicyclic alkane derivatives as the biaryl substituted of nicotinic acetylcholine receptor activity modulators ABBOTT LAB 2010-12-22 CN disclosed
CN-101918409-A The diazabicycloalkane derivatives of biaryl substituted ABBOTT LAB 2010-12-15 CN disclosed
CN-101918358-A Novel vitamin D receptor activators and methods of manufacture ABBOTT LAB 2010-12-15 CN disclosed
CN-101309922-A Amino-aza-adamantane derivatives and methods of use ABBOTT LAB (US) 2008-11-19 CN disclosed