SCHEMBL2479592

SCHEMBL2479592

Clc1ccc([CH]c2ccccc2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
G6PC1 P35575 1/20 0.46
NPFFR2 Q9Y5X5 2/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CHAT P28329 1/20 0.40
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
IDO2 Q6ZQW0 1/20 0.39
AHR P35869 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.37
GPR183 P32249 1/20 0.37
PYGL P06737 1/20 0.37
IGF1R P08069 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
KDM4A O75164 1/20 0.36
KDM4B O94953 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3298582 0.88 ALDH1A1 (0.64) ALDH1A1G6PC1NPFFR2KMT2ANPSR1
SCHEMBL19036493 0.82 CHAT (0.58) ALDH1A1G6PC1CHATPYGLKDM4A
SCHEMBL10712182 0.82 CHAT (0.58) ALDH1A1G6PC1CHATPYGLKDM4A
SCHEMBL10712185 0.82 CHAT (0.58) ALDH1A1G6PC1CHATPYGLKDM4A
SCHEMBL2357484 0.77 ALDH1A1 (0.50) ALDH1A1KMT2ACHATLMNATSHR
SCHEMBL439444 0.75 G6PD (0.54) G6PC1LMNATSHRIDO1TDO2
SCHEMBL3301775 0.74 CHRM5 (0.56) ALDH1A1KMT2ACHATTSHRMAPT
SCHEMBL1302 0.74 ALDH1A1 (0.53) ALDH1A1KMT2ACHATLMNATSHR
SCHEMBL11409587 0.72 ALDH1A1 (0.56) ALDH1A1G6PC1NPFFR2KMT2ANPSR1
SCHEMBL10973255 0.72 ALDH1A1 (0.64) ALDH1A1NPFFR2KMT2ANPSR1CHAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8492384-B2 Imidazolylalkylcarbonyl derivatives as calcium channel modulators and preparation method thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2013-07-23 US claimed
EP-2231613-B1 MONTELUKAST BENZHYDRYL PIPERAZINE SALTS AND PROCESS FOR PREPARATION THEREOF TORRENT PHARMACEUTICALS LTD (IN) 2011-10-12 EP claimed
US-20090325979-A1 NOVEL IMIDAZOLYLALKYLCARBONYL DERIVATIVES AS CALCIUM CHANNEL MODULATORS AND PREPARATION METHOD THEREOF KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-12-31 US claimed
US-8492384-B2 Imidazolylalkylcarbonyl derivatives as calcium channel modulators and preparation method thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2013-07-23 US disclosed
US-8299072-B2 Pyrazolylmethylamine compounds as calcium channel modulators and preparation method thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2012-10-30 US disclosed
US-20100094006-A1 NOVEL PYRAZOLYLMETHYLAMINE COMPOUNDS AS CALCIUM CHANNEL MODULATORS AND PREPARATION METHOD THEREOF KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2010-04-15 US disclosed
US-20090325979-A1 NOVEL IMIDAZOLYLALKYLCARBONYL DERIVATIVES AS CALCIUM CHANNEL MODULATORS AND PREPARATION METHOD THEREOF KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-12-31 US disclosed
WO-2000069893-A1 GLYCOPEPTIDE ANTIBACTERIAL COMPOUNDS, COMPOSITIONS CONTAINING SAME AND METHODS OF USING SAME MERCK & CO., INC. (US) 2000-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325979-A1 NOVEL IMIDAZOLYLALKYLCARBONYL DERIVATIVES AS CALCIUM CHANNEL MODULATORS AND PREPARATION METHOD THEREOF CACNA1B, CACNA1C, ORAI1 ALDH1A1 3972/4885G6PC1 1620/4885NPFFR2 1192/4885
US-20100094006-A1 NOVEL PYRAZOLYLMETHYLAMINE COMPOUNDS AS CALCIUM CHANNEL MODULATORS AND PREPARATION METHOD THEREOF CACNA1I, CACNA1C, ORAI1 ALDH1A1 4048/4885G6PC1 1679/4885NPFFR2 941/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.