SCHEMBL24802441

SCHEMBL24802441

Cc1cnc(O)c(CCN(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.40
HTR2A P28223 5/20 0.40
HTR2C P28335 5/20 0.40
HTR2B P41595 3/20 0.40
SLC6A4 P31645 1/20 0.40
HTR7 P34969 2/20 0.37
HTR6 P50406 2/20 0.36
DRD1 P21728 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR1E P28566 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
DRD3 P35462 1/20 0.36
HTR5A P47898 1/20 0.36
TAAR1 Q96RJ0 3/20 0.34
MDM2 Q00987 1/20 0.34
MPO P05164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24802482 0.76 SLC13A5 (0.49) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL25795552 0.75 NOS3 (0.39)
SCHEMBL24802437 0.72 GAA (0.35) HTR2B
SCHEMBL25246536 0.72 HTR6 (0.48) HTR1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL30566012 0.72 HTR6 (0.48) HTR1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL21459479 0.71 HTR7 (0.37) HTR1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL10949866 0.70 AMY1A (0.52) HTR1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL30148591 0.69 HTR2A (0.49) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL29038139 0.68 HTR2A (0.40) HTR1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL21459468 0.66 HTR2A (0.41) HTR1AHTR2AHTR2CHTR2BSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed