SCHEMBL2481589

SCHEMBL2481589

CC(C)(NC(=O)[C@@]1(c2ccc(F)cc2)C[C@H]1CO)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.41
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
SLC6A2 P23975 3/20 0.40
TACR1 P25103 1/20 0.39
TACR3 P29371 5/20 0.39
SLC6A4 P31645 2/20 0.39
SSTR4 P31391 1/20 0.38
OPRL1 P41146 1/20 0.37
MAOB P27338 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2477280 0.92 SLC6A2 (0.47) SLC6A2SLC6A4SSTR4MAOB
SCHEMBL2477910 0.88 TMEM97 (0.42) SLC6A2
SCHEMBL2476151 0.88 TACR3 (0.40) RORCCNR1CNR2SLC6A2TACR1
SCHEMBL2481591 0.83 TACR3 (0.41) TACR1TACR3SLC6A4
SCHEMBL5791908 0.75 HSD11B1 (0.44) MAOB
SCHEMBL3744181 0.75 HSD11B1 (0.44) MAOB
SCHEMBL5788833 0.73 SIGMAR1 (0.46)
N-Benzylmethylamine SCHEMBL2477939 0.73 SLC6A4 (0.44) RORCSLC6A2TACR3SLC6A4OPRL1
SCHEMBL17735432 0.71 SLC6A4 (0.56) SLC6A2SLC6A4OPRL1OPRM1
SCHEMBL2477938 0.71 TACR3 (0.60) SLC6A2TACR3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP disclosed