SCHEMBL2476151

SCHEMBL2476151

CC(C)(NC(=O)[C@@]1(c2ccc(F)c(F)c2)C[C@H]1CO)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 2/20 0.40
VNN1 O95497 1/20 0.38
SSTR4 P31391 1/20 0.36
CCR2 P41597 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 1/20 0.34
TACR1 P25103 1/20 0.34
RORC P51449 1/20 0.34
KCNN4 O15554 1/20 0.34
IMPDH2 P12268 1/20 0.34
CNR2 P34972 4/20 0.33
CNR1 P21554 3/20 0.33
PPARG P37231 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ACKR3 P25106 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2481589 0.88 RORC (0.41) TACR3SSTR4SLC6A2SLC6A4TACR1
SCHEMBL2477280 0.86 SLC6A2 (0.47) SSTR4SLC6A2SLC6A4
SCHEMBL2477910 0.85 TMEM97 (0.42) SLC6A2
SCHEMBL2481591 0.85 TACR3 (0.41) TACR3SLC6A4TACR1
SCHEMBL3743997 0.77 CCR2 (0.43) TACR3CCR2SLC6A2SLC6A4
SCHEMBL6023197 0.77 CCR2 (0.43) TACR3CCR2SLC6A2SLC6A4
SCHEMBL5792435 0.75 SIGMAR1 (0.42) CCR2
N-Benzylmethylamine SCHEMBL2477949 0.75 TACR3 (0.40) TACR3CCR2SLC6A2SLC6A4
N-Benzylmethylamine SCHEMBL5792207 0.75 TACR3 (0.40) TACR3CCR2SLC6A2SLC6A4
SCHEMBL5792205 0.72 TACR3 (0.59) TACR3TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP disclosed