SCHEMBL2477910

SCHEMBL2477910

CC(C)(NC(=O)[C@@]1(c2ccc(Cl)cc2)C[C@H]1CO)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
SLC6A2 P23975 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2477280 0.92 SLC6A2 (0.47) SLC6A2
SCHEMBL2481589 0.88 RORC (0.41) SLC6A2
SCHEMBL2481591 0.88 TACR3 (0.41)
SCHEMBL2476151 0.85 TACR3 (0.40) SLC6A2
SCHEMBL5789157 0.75 TMEM97 (0.42) TMEM97SIGMAR1
SCHEMBL3742011 0.75 TMEM97 (0.42) TMEM97SIGMAR1
SCHEMBL5791992 0.73 SIGMAR1 (0.58) TMEM97SIGMAR1
N-Benzylmethylamine SCHEMBL2477549 0.73 SLC6A4 (0.44) TMEM97SIGMAR1SLC6A2
SCHEMBL17735432 0.71 SLC6A4 (0.56) SLC6A2
SCHEMBL2477546 0.71 TACR3 (0.55) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656349-B1 CYCLOPROPYL DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS LUNDBECK & CO AS H (DK) 2011-10-12 EP disclosed