SCHEMBL2482403

SCHEMBL2482403

CN(Cc1cccnc1)C(=O)CCCSc1cccc(O)c1.COc1ccc(SCCCC(=O)N(C)Cc2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.46
LMNA P02545 4/20 0.43
ALDH1A1 P00352 3/20 0.43
CLK1 P49759 1/20 0.43
MAPK1 P28482 1/20 0.43
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 2/20 0.41
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.39
HSD17B2 P37059 1/20 0.39
LRRK2 Q5S007 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2485825 0.92 LMNA (0.47) PDK1LMNAKMT2ASMN1; SMN2HTT
SCHEMBL2487605 0.92 PDK1 (0.42) PDK1LMNAALDH1A1CLK1MAPK1
SCHEMBL416236 0.89 CLK1 (0.49) PDK1LMNAALDH1A1CLK1MAPK1
SCHEMBL417568 0.89 RIPK1 (0.46) PDK1LMNAALDH1A1CLK1KMT2A
SCHEMBL416207 0.83 MAPK1 (0.60) LMNAALDH1A1MAPK1MAPTKMT2A
SCHEMBL418540 0.83 NPC1 (0.55) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL418243 0.82 RIPK1 (0.49) PDK1LMNAALDH1A1MAPTPOLB
SCHEMBL2484074 0.82 LMNA (0.47) LMNAALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL2482708 0.78 TSHR (0.54) LMNAALDH1A1MAPK1MAPTKMT2A
SCHEMBL412372 0.78 ALDH1A1 (0.53) LMNAALDH1A1MAPK1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376431-A1 NOVEL SUBSTITUTED ARYL DERIVATIVES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTICAL USES AS ANTI-HIV AGENTS LABORATOIRE BIODIM (FR) 2011-10-19 EP disclosed
WO-2010066847-A1 NOVEL SUBSTITUTED ARYL DERIVATIVES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTICAL USES AS ANTI-HIV AGENTS CELLVIR (FR) 2010-06-17 WO disclosed