SCHEMBL2483148

SCHEMBL2483148

NS(=O)(=O)c1ccc2nc(C(=O)Nc3ccccc3)cn2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.62
RAB9A P51151 3/20 0.62
CYP2C9 P11712 1/20 0.58
NR4A2 P43354 1/20 0.58
CA1 P00915 5/20 0.53
CA2 P00918 5/20 0.53
CA12 O43570 3/20 0.50
CA9 Q16790 3/20 0.50
MAPT P10636 6/20 0.47
KMT2A Q03164 3/20 0.46
POLB P06746 3/20 0.46
MEN1 O00255 2/20 0.46
PSMD14 O00487 1/20 0.46
RECQL P46063 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
SAE1 Q9UBE0 1/20 0.46
UBA2 Q9UBT2 1/20 0.46
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2484415 0.88 NPC1 (0.62) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2483734 0.85 NPC1 (0.60) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2485145 0.84 RAB9A (0.58) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2485532 0.82 RAB9A (0.68) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2485519 0.82 RAB9A (0.68) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL21033165 0.81 PTGS1 (0.51) CA1CA2CA12CA9KMT2A
SCHEMBL3367654 0.80 RAB9A (0.70) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3368461 0.80 NPC1 (0.70) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3367363 0.80 NPC1 (0.65) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3367614 0.79 RAB9A (0.72) NPC1RAB9ACYP2C9NR4A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225245-B1 N-phenyl-imidazo(1,2-a)pyridine-2-carboxamide compounds, preparation thereof and therapeutic application thereof SANOFI SA (FR) 2011-10-19 EP claimed
US-20100317620-A1 N-PHENYLIMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE COMPOUNDS, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-12-16 US claimed
EP-2225245-B1 N-phenyl-imidazo(1,2-a)pyridine-2-carboxamide compounds, preparation thereof and therapeutic application thereof SANOFI SA (FR) 2011-10-19 EP disclosed
US-20100317620-A1 N-PHENYLIMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE COMPOUNDS, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100317620-A1 N-PHENYLIMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE COMPOUNDS, PREPARATION AND THERAPEUTIC USE THEREOF GLS, REN, XDH NPC1 595/4885RAB9A 1438/4885CYP2C9 806/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.