SCHEMBL2484415

SCHEMBL2484415

CS(=O)(=O)c1ccc2nc(C(=O)Nc3ccccc3)cn2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.62
RAB9A P51151 4/20 0.62
CYP2C9 P11712 1/20 0.58
NR4A2 P43354 1/20 0.58
MAPT P10636 2/20 0.47
POLB P06746 1/20 0.46
KDM4E B2RXH2 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PRKDC P78527 1/20 0.45
ATR Q13535 1/20 0.45
EGLN1 Q9GZT9 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HSP90AA1 P07900 1/20 0.44
KMT2A Q03164 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
CCNB2 O95067 2/20 0.44
CCNE2 O96020 2/20 0.44
CDK1 P06493 2/20 0.44
CDK4 P11802 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2483734 0.88 NPC1 (0.60) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2483148 0.88 NPC1 (0.62) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2485145 0.87 RAB9A (0.58) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3368461 0.83 NPC1 (0.70) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2485532 0.82 RAB9A (0.68) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3365483 0.81 NPC1 (0.67) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3367654 0.80 RAB9A (0.70) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL2487512 0.80 NPC1 (0.62) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3365520 0.80 NPC1 (0.65) NPC1RAB9ACYP2C9NR4A2MAPT
SCHEMBL3371083 0.80 NPC1 (0.65) NPC1RAB9ACYP2C9NR4A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225245-B1 N-phenyl-imidazo(1,2-a)pyridine-2-carboxamide compounds, preparation thereof and therapeutic application thereof SANOFI SA (FR) 2011-10-19 EP claimed
US-20100317620-A1 N-PHENYLIMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE COMPOUNDS, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-12-16 US claimed
EP-2225245-B1 N-phenyl-imidazo(1,2-a)pyridine-2-carboxamide compounds, preparation thereof and therapeutic application thereof SANOFI SA (FR) 2011-10-19 EP disclosed
US-20100317620-A1 N-PHENYLIMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE COMPOUNDS, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100317620-A1 N-PHENYLIMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE COMPOUNDS, PREPARATION AND THERAPEUTIC USE THEREOF GLS, REN, XDH NPC1 595/4885RAB9A 1438/4885CYP2C9 806/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.