SCHEMBL2483598

SCHEMBL2483598

CC(C)Oc1ccccc1CN(C)C(=O)CCCSc1ccc(O)cc1.CN(Cc1ccccc1Cl)C(=O)CCCSc1ccc(F)cc1.COC(=O)c1ccc(SCCCC(=O)NCCc2ccccc2OC)cc1.COc1ccc(SCCCC(=O)N(C)Cc2ccccc2OC)cc1.COc1ccccc1CN(C)C(=O)CCCSc1cnc2ccccc2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.33
HCRTR2 O43614 1/20 0.31
ALDH1A1 P00352 2/20 0.31
MAPT P10636 2/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
PPARG P37231 1/20 0.31
ADRB2 P07550 1/20 0.31
TP53 P04637 1/20 0.30
NPC1 O15118 2/20 0.30
LMNA P02545 2/20 0.30
RAB9A P51151 2/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
USP5 P45974 1/20 0.30
BRAP Q7Z569 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
USP16 Q9Y5T5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487639 0.85 HTR7 (0.34) KMT2A
SCHEMBL2482378 0.85
SCHEMBL417292 0.76 TP53 (0.37) RXFP1ALDH1A1PPARGTP53NPC1
SCHEMBL414416 0.72 ACHE (0.48) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL417291 0.70 L3MBTL1 (0.39) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL418468 0.70 BCHE (0.43) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL414461 0.70 ALDH1A1 (0.52) ALDH1A1ADRB2NPC1RAB9AKMT2A
SCHEMBL414460 0.70 ACHE (0.51) ALDH1A1LMNARAB9AKMT2ATDP1
SCHEMBL416337 0.70 BCHE (0.43) ALDH1A1KMT2ATDP1
SCHEMBL416610 0.69 NPC1 (0.45) ALDH1A1NPC1LMNARAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376431-A1 NOVEL SUBSTITUTED ARYL DERIVATIVES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTICAL USES AS ANTI-HIV AGENTS LABORATOIRE BIODIM (FR) 2011-10-19 EP disclosed
WO-2010066847-A1 NOVEL SUBSTITUTED ARYL DERIVATIVES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTICAL USES AS ANTI-HIV AGENTS CELLVIR (FR) 2010-06-17 WO disclosed