SCHEMBL2487639

SCHEMBL2487639

CN(Cc1ccccc1Cl)C(=O)CCCSc1ccc(F)cc1.CN(Cc1ccccc1O)C(=O)CCCSc1ccc(F)cc1.CN1CCN(c2ccccc2CN(C)C(=O)CCCSc2ccc(O)cc2)CC1.COC(=O)c1ccc(SCCCC(=O)NCCc2ccccc2OC)cc1.COc1ccccc1CN(C)C(=O)CCCSc1cnc2ccccc2n1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 15/20 0.34
HTR1A P08908 10/20 0.34
KMT2A Q03164 1/20 0.34
HTR2C P28335 4/20 0.33
HTR2A P28223 3/20 0.33
HTR1D P28221 2/20 0.33
HTR1B P28222 2/20 0.33
HTR5A P47898 2/20 0.33
HTR6 P50406 2/20 0.33
DRD2 P14416 3/20 0.33
DRD3 P35462 2/20 0.33
SLC2A1 P11166 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2483598 0.85 RXFP1 (0.33) KMT2A
SCHEMBL2482378 0.77
SCHEMBL416317 0.70 NCF1 (0.37) HTR7HTR1AKMT2AHTR2CHTR2A
SCHEMBL414416 0.70 ACHE (0.48) KMT2A
SCHEMBL2487851 0.69 SMN1; SMN2 (0.37) HTR7HTR1AKMT2ADRD2DRD3
SCHEMBL414461 0.68 ALDH1A1 (0.52) KMT2A
SCHEMBL414460 0.68 ACHE (0.51) KMT2A
SCHEMBL2481990 0.66 DRD2 (0.34) HTR1AKMT2AHTR2ADRD2DRD3
SCHEMBL412451 0.65 ACHE (0.54) KMT2A
SCHEMBL413455 0.65 ACHE (0.54) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376431-A1 NOVEL SUBSTITUTED ARYL DERIVATIVES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTICAL USES AS ANTI-HIV AGENTS LABORATOIRE BIODIM (FR) 2011-10-19 EP claimed
WO-2010066847-A1 NOVEL SUBSTITUTED ARYL DERIVATIVES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTICAL USES AS ANTI-HIV AGENTS CELLVIR (FR) 2010-06-17 WO claimed