Oxapium

Oxapium

SCHEMBL24857

C[N+]1(CC2COC(c3ccccc3)(C3CCCCC3)O2)CCCCC1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTDSP1 Q9GZU7 4/20 0.47
PABPC1 P11940 1/20 0.47
APOBEC3A P31941 2/20 0.42
APOBEC3G Q9HC16 2/20 0.42
KMT2A Q03164 1/20 0.42
CHRM2 P08172 10/20 0.41
CHRM4 P08173 10/20 0.41
CHRM5 P08912 10/20 0.41
CHRM1 P11229 10/20 0.41
CHRM3 P20309 10/20 0.41
GRIN1 Q05586 2/20 0.39
GRIN2A Q12879 2/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxapium SCHEMBL1316687 0.99 CTDSP1 (0.49) CTDSP1PABPC1APOBEC3AAPOBEC3GKMT2A
SCHEMBL27721335 0.79 GRIN1 (0.44) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11259848 0.75 HTR1A (0.49) CHRM2CHRM4CHRM5CHRM1CHRM3
Hydrochloric Acid SCHEMBL29449197 0.74 HTR1A (0.48) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL14039627 0.72 CHRM2 (0.43) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL10807843 0.72 GAA (0.49) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL10807846 0.70 CHRM2 (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL19420724 0.66 CTDSP1 (0.97) CTDSP1PABPC1APOBEC3AAPOBEC3GKMT2A
SCHEMBL19420729 0.66 CTDSP1 (0.97) CTDSP1PABPC1APOBEC3AAPOBEC3GKMT2A
SCHEMBL28274789 0.63 CYP3A4 (0.38) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 681 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119630804-A Batch process for enzymatic modification of lipids 邦吉SA公司 2025-03-14 CN claimed
CN-118806672-A Sleeping mask and preparation method thereof 上海珈制化妆品有限公司 2024-10-22 CN claimed
US-20240229089-A1 A process for enzymatic synthesis of amides from amines and carboxylic acids or esters XP CHEMISTRIES AB (SE) 2024-07-11 US claimed
EP-4308714-A1 A PROCESS FOR ENZYMATIC SYNTHESIS OF AMIDES FROM AMINES AND CARBOXYLIC ACIDS OR ESTERS XP Chemistries AB (SE) 2024-01-24 EP claimed
CN-117305391-A Method for regulating molecular weight of dextran by enzymolysis 广西民族大学 2023-12-29 CN claimed
CN-116490160-A A mixture containing 1, 2-alkanediol 西姆莱斯股份公司 2023-07-25 CN claimed
WO-2022229314-A1 A PROCESS FOR ENZYMATIC SYNTHESIS OF AMIDES FROM AMINES AND CARBOXYLIC ACIDS OR ESTERS XP CHEMISTRIES AB (SE) 2022-11-03 WO claimed
EP-4077697-A1 CARBOXYLIC ACID ESTERS OF XYLITOL AND PROCESS FOR ENZYMATICALLY PREPARING SAME Evonik Operations GmbH (DE) 2022-10-26 EP claimed
EP-4077696-A1 PROCESS FOR ENZYMATICALLY PREPARING SUGAR ESTERS AND/OR SUGAR ALCOHOL ESTERS Evonik Operations GmbH (DE) 2022-10-26 EP claimed
EP-4077698-A1 SORBITAN ESTERS AND PROCESS FOR ENZYMATICALLY PREPARING SAME Evonik Operations GmbH (DE) 2022-10-26 EP claimed
CN-101121708-B Method for synthesizing oxapium iodide and analogue thereof XIAOXIANG LI 2010-12-15 CN claimed
EP-1879578-A4 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV PHARMACEUTICAL INC (US) 2009-05-13 EP claimed
CN-101121708-A Method for synthesizing oxapium iodide and analogue thereof XIAOXIANG LI (CN) 2008-02-13 CN claimed
EP-1879578-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV Pharmaceutical Inc. (US) 2008-01-23 EP claimed
WO-2006102029-A9 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV PHARMACEUTICAL INC (US) 2006-12-07 WO claimed
WO-2006102029-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV PHARMACEUTICAL, INC. (US) 2006-09-28 WO claimed
WO-2006075908-A1 WATER TREATMENT DEVICE WHICH DEACTIVATES ELECTROMAGNETIC RADIATION DEL TORO PADILLA BEATRIZ ANGEL (MX) 2006-07-20 WO claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5811547-A Method for inducing crystalline state transition in medicinal substance NIPPON SHINYAJU CO., LTD. (JP) 1998-09-22 US claimed