SCHEMBL24875987

SCHEMBL24875987

COc1nc2ccc(C[PH](c3ccccc3)(c3ccccc3)c3ccccc3)cc2nc1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NQO2 P16083 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NR1I3 Q14994 2/20 0.35
MAPK1 P28482 1/20 0.35
HRH4 Q9H3N8 3/20 0.34
HPGD P15428 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
VDR P11473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16541886 0.73 CA2 (0.53) KDM4EMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL2145470 0.73 GAA (0.57) MEN1KMT2AALDH1A1LMNAL3MBTL1
SCHEMBL3275902 0.73 MEN1 (0.39) KDM4EMEN1KMT2ANQO2NPC1
SCHEMBL24875977 0.72 KDM4E (0.38) KDM4EMEN1KMT2ANQO2NPC1
Bromide SCHEMBL16180801 0.72 CA2 (0.52) KDM4EMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL13403262 0.71 KDM1A (0.46) KDM4EMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL7819280 0.71 LTA4H (0.57) NPC1RAB9ATP53
SCHEMBL24635162 0.71 NCF1 (0.49) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL5973660 0.70 MAOB (0.57) KDM4EALDH1A1CYP1A2
SCHEMBL9088704 0.70 GAA (0.54) KDM4EMEN1KMT2ARAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023280970-A1 INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2023-01-12 WO disclosed