SCHEMBL2488367

SCHEMBL2488367

CC(C)(C)c1ccc(Oc2ccc3cc(C(C)(C)N)ccc3c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.56
NPC1 O15118 3/20 0.56
HPGD P15428 3/20 0.56
MAPT P10636 3/20 0.56
ALDH1A1 P00352 2/20 0.56
MAPK1 P28482 1/20 0.56
BCHE P06276 4/20 0.43
ACHE P22303 4/20 0.43
KDM4E B2RXH2 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
ADAMTS5 Q9UNA0 2/20 0.39
FGFR2 P21802 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2452091 0.88 RAB9A (0.43) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2455599 0.85 RAB9A (0.51) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2451911 0.85 RAB9A (0.51) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2457235 0.83 NPC1 (0.42) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2449570 0.83 MAPT (0.45) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2452036 0.81 RAB9A (0.36) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2449524 0.81 SOS1 (0.44) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2452741 0.80 NPC1 (0.36) RAB9ANPC1HPGDMAPTALDH1A1
SCHEMBL2449797 0.79 AR (0.42) MAPTALDH1A1POLBGAACYP1A2
SCHEMBL2448045 0.79 KIF11 (0.50) MAPTALDH1A1KDM4EPOLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364088-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS Biogen Idec MA Inc. (US) 2011-09-14 EP disclosed
WO-2010051030-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS BIOGEN IDEC MA INC. (US) 2010-05-06 WO disclosed