SCHEMBL2452741

SCHEMBL2452741

CC(C)Cc1ccc(Oc2ccc3cc(C(C)(C)N)ccc3c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
KDM4C Q9H3R0 1/20 0.35
SLC6A4 P31645 1/20 0.35
ST14 Q9Y5Y6 1/20 0.34
FFAR1 O14842 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2449767 0.89 PTGS2 (0.35) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL2449764 0.89 PTGS2 (0.35) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL2457235 0.84 NPC1 (0.42) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL2488367 0.80 RAB9A (0.56) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL2452091 0.79 RAB9A (0.43) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL13719230 0.77 ALDH1A1 (0.46) ALDH1A1FFAR1
SCHEMBL4575613 0.76 SLC6A4 (0.48) TSHRSLC6A4ST14HTR2A
SCHEMBL2448201 0.74 PTGS1 (0.39) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL2449570 0.74 MAPT (0.45) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL2452036 0.73 RAB9A (0.36) NPC1MAPTRAB9AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364088-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS Biogen Idec MA Inc. (US) 2011-09-14 EP disclosed
WO-2010051030-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS BIOGEN IDEC MA INC. (US) 2010-05-06 WO disclosed