SCHEMBL2488979

SCHEMBL2488979

O=C(O)Oc1cn(Cc2ccc(-c3ccc4c(c3)OCCO4)cc2F)c2c(F)ccc(F)c2c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 4/20 0.39
NAAA Q02083 1/20 0.36
PKM P14618 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
CD274 Q9NZQ7 2/20 0.34
MAPT P10636 4/20 0.34
TP53 P04637 3/20 0.34
RAB9A P51151 3/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
HTT P42858 2/20 0.33
HSD17B10 Q99714 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2488977 0.86 CHRM1 (0.55) CHRM1NAAAPKMTDP1MAPT
SCHEMBL2486084 0.86 CHRM1 (0.53) CHRM1MAPTTP53P2RX7
SCHEMBL2492208 0.82 CHRM1 (0.41) CHRM1
SCHEMBL2488348 0.81 CHRM1 (0.40) CHRM1
SCHEMBL2492205 0.81 CHRM1 (0.41) CHRM1
SCHEMBL2488465 0.80 CHRM1 (0.41) CHRM1P2RX7
SCHEMBL2487909 0.80 CHRM1 (0.43) CHRM1P2RX7
SCHEMBL2491881 0.79 ERN1 (0.42) CHRM1
SCHEMBL2488025 0.79 CHRM1 (0.41) CHRM1RAB9ANPC1POLBGAA
SCHEMBL2487494 0.78 CHRM1 (0.40) CHRM1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037739-B1 BENZYL-SUBSTITUTED QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2011-10-26 EP claimed