SCHEMBL24891766

SCHEMBL24891766

COc1cc(NC(=O)c2ccc(C(=O)Nc3ccc(CNC(=N)N)cc3)cc2)ccc1C1=CCN(C(=N)N)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 5/20 0.47
NAMPT P43490 4/20 0.47
MAPT P10636 2/20 0.42
USP2 O75604 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ABCB1 P08183 2/20 0.41
ABCG2 Q9UNQ0 2/20 0.41
KMT2A Q03164 2/20 0.40
ROCK2 O75116 2/20 0.40
CYP3A4 P08684 1/20 0.40
HTR1D P28221 1/20 0.40
SLC6A4 P31645 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30181059 0.90 TMPRSS2 (0.48) TMPRSS2NAMPTMAPTLMNAHTR1D
SCHEMBL29802915 0.89 TMPRSS2 (0.49) TMPRSS2NAMPTMAPTLMNAHTR1D
SCHEMBL24669441 0.88 TMPRSS2 (0.53) TMPRSS2NAMPTMAPTUSP2ALDH1A1
SCHEMBL29802955 0.87 TMPRSS2 (0.45) TMPRSS2NAMPTMAPTHDAC1TP53
SCHEMBL24671223 0.87 TMPRSS2 (0.45) TMPRSS2NAMPTMAPTHDAC1TP53
SCHEMBL24891726 0.87 ALDH1A1 (0.43) TMPRSS2NAMPTMAPTALDH1A1HPGD
SCHEMBL24891885 0.86 TMPRSS2 (0.45) TMPRSS2NAMPTMAPTALDH1A1HPGD
SCHEMBL24669387 0.86 TMPRSS2 (0.45) TMPRSS2NAMPTMAPTALDH1A1HPGD
SCHEMBL24671334 0.85 TMPRSS2 (0.43) TMPRSS2NAMPTMAPTLMNATP53
SCHEMBL24670178 0.84 TMPRSS2 (0.52) TMPRSS2NAMPTMAPTUSP2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO claimed
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed