SCHEMBL24901460

SCHEMBL24901460

CCOC(=O)C(F)(F)Oc1ccc(Br)c(C)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.37
PIN1 Q13526 1/20 0.36
EPHX2 P34913 1/20 0.36
FBP1 P09467 3/20 0.36
CYP1A2 P05177 2/20 0.35
ABCB11 O95342 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
HTR2A P28223 1/20 0.35
PMP22 Q01453 1/20 0.35
PPARA Q07869 1/20 0.35
POLB P06746 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
LMNA P02545 3/20 0.34
CES2 O00748 1/20 0.34
ACHE P22303 1/20 0.34
CES1 P23141 1/20 0.34
HTT P42858 1/20 0.34
PKM P14618 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15094227 0.78 PIN1 (0.45) MAPTPIN1EPHX2FBP1TSHR
SCHEMBL22123345 0.77 FBP1 (0.50) PIN1FBP1CYP1A2ABCB11CYP3A4
SCHEMBL24901468 0.76 KMT2A (0.43) FBP1CYP1A2TSHRPOLBNPSR1
SCHEMBL24901718 0.76 KCNA3 (0.34) MAPTEPHX2FBP1CYP1A2ABCB11
SCHEMBL31697054 0.75 PDE2A (0.34) EPHX2
SCHEMBL22207999 0.75 PDE2A (0.34) EPHX2
SCHEMBL24901456 0.75
SCHEMBL24901695 0.74 ALDH1A1 (0.49) FBP1CYP1A2ABCB11CYP3A4TSHR
SCHEMBL24901453 0.74 ALDH1A1 (0.42) MAPTCYP1A2TSHRPOLBLMNA
SCHEMBL24901458 0.73 FBP1 (0.46) MAPTEPHX2FBP1CYP1A2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023286768-A1 HYDROGENATED QUINOXALINES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2023-01-19 WO disclosed