SCHEMBL249020

SCHEMBL249020

C=CCc1cccc2c1c(C=O)c(C)n2C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
KMT2A Q03164 8/20 0.35
MEN1 O00255 7/20 0.35
USP2 O75604 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 2/20 0.34
PSMD14 O00487 1/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PKM P14618 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250231 0.72 GABRA1 (0.36) HTTALDH1A1SMN1; SMN2GABRA1GABRB2
SCHEMBL3083235 0.69 GABRA1 (0.50) ALDH1A1GABRA1GABRB2KMT2AMEN1
SCHEMBL8791921 0.69 GABRA1 (0.43) ALDH1A1GABRA1GABRB2KMT2AMEN1
SCHEMBL166586 0.66 GABRA1 (0.52) ALDH1A1GABRA1GABRB2KMT2AMEN1
Acetic Acid SCHEMBL27930745 0.65 GABRA1 (0.43) HTTALDH1A1SMN1; SMN2GABRA1GABRB2
SCHEMBL13265468 0.64 GABRA1 (0.44) HTTALDH1A1SMN1; SMN2GABRA1GABRB2
Acetic Acid SCHEMBL9771555 0.64 GABRA1 (0.63) HTTALDH1A1SMN1; SMN2GABRA1GABRB2
SCHEMBL7369721 0.63 MRGPRX4 (0.45) HTTALDH1A1SMN1; SMN2GABRA1GABRB2
SCHEMBL5226691 0.62 ALDH1A1 (0.57) ALDH1A1GABRA1GABRB2KMT2AMEN1
SCHEMBL10961297 0.62 AKR1C3 (0.46) ALDH1A1SMN1; SMN2GABRA1GABRB2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001308-A9 METHOD FOR SYNTHESIZING ERGOLINE ALKALOIDS FROM INDOLIC BICYCLIC COMPOUNDS BY DOUBLE CYCLIZATION, RESULTING MATERIALS, AND INTERMEDIATE MATERIALS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-03-22 WO disclosed
WO-2012001308-A1 METHOD FOR SYNTHESIZING ERGOLINE ALKALOIDS FROM INDOLIC BICYCLIC COMPOUNDS BY DOUBLE CYCLIZATION, RESULTING MATERIALS, AND INTERMEDIATE MATERIALS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-01-05 WO disclosed