SCHEMBL250231

SCHEMBL250231

C=CCc1cccc2c1c(C=O)cn2C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
MEN1 O00255 6/20 0.34
KMT2A Q03164 6/20 0.34
KDM4E B2RXH2 4/20 0.33
HTT P42858 4/20 0.33
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
MAPT P10636 2/20 0.33
ALOX12 P18054 1/20 0.33
ALDH1A1 P00352 3/20 0.33
PKM P14618 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
TDP1 Q9NUW8 2/20 0.31
CASP3 P42574 1/20 0.31
RECQL P46063 1/20 0.31
CASP7 P55210 1/20 0.31
MTOR P42345 1/20 0.31
RAB9A P51151 1/20 0.31
POLB P06746 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805996 0.82 L3MBTL1 (0.42) GABRA1GABRB2MEN1KMT2AALDH1A1
SCHEMBL249361 0.80 ERN1 (0.33) MEN1KMT2ALMNAALDH1A1L3MBTL1
SCHEMBL20503064 0.76 CYP2A6 (0.41) MEN1KMT2AKDM4EALDH1A1L3MBTL1
SCHEMBL15901985 0.76 ALDH1A1 (0.36) MEN1KMT2AKDM4EHTTSMN1; SMN2
SCHEMBL15902473 0.76 ALDH1A1 (0.39) MEN1KMT2AALDH1A1L3MBTL1TDP1
SCHEMBL20503055 0.72 RORC (0.40)
SCHEMBL249020 0.72 HTT (0.37) GABRA1GABRB2MEN1KMT2AKDM4E
SCHEMBL22126563 0.70 NOTUM (0.36) ALDH1A1PKML3MBTL1TDP1CASP3
SCHEMBL5736785 0.68 ALDH1A1 (0.56) MEN1KMT2AKDM4EHTTLMNA
SCHEMBL30234384 0.68 ALDH1A1 (0.56) MEN1KMT2AKDM4EHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001308-A9 METHOD FOR SYNTHESIZING ERGOLINE ALKALOIDS FROM INDOLIC BICYCLIC COMPOUNDS BY DOUBLE CYCLIZATION, RESULTING MATERIALS, AND INTERMEDIATE MATERIALS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-03-22 WO disclosed
WO-2012001308-A1 METHOD FOR SYNTHESIZING ERGOLINE ALKALOIDS FROM INDOLIC BICYCLIC COMPOUNDS BY DOUBLE CYCLIZATION, RESULTING MATERIALS, AND INTERMEDIATE MATERIALS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-01-05 WO disclosed