SCHEMBL24920436

SCHEMBL24920436

COCCCN1CCC(CN2CCC3(CC2)CN(C)C3)CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
HTR4 Q13639 4/20 0.33
CYP2D6 P10635 2/20 0.33
CYP3A4 P08684 1/20 0.33
HRH3 Q9Y5N1 5/20 0.33
HRH1 P35367 2/20 0.33
HRH2 P25021 1/20 0.33
CYP1A2 P05177 1/20 0.33
ALOX15 P16050 1/20 0.33
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
ACHE P22303 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29325624 0.90 HRH1 (0.36) MEN1CYP2D6HRH3HRH1HRH2
SCHEMBL19977411 0.87 DRD2 (0.37) MEN1HTR4CYP2D6HRH3CYP1A2
SCHEMBL24920438 0.84 DRD2 (0.34) MEN1HTR4CYP2D6HRH3CYP1A2
SCHEMBL24920953 0.83 SIGMAR1 (0.37) SIGMAR1
SCHEMBL24920944 0.83 SIGMAR1 (0.37) SIGMAR1
SCHEMBL24921699 0.81 DRD2 (0.34) MEN1HTR4CYP2D6HRH3CYP1A2
SCHEMBL22565121 0.80 NCF1 (0.41) SIGMAR1ACHEOPRM1OPRK1OPRL1
SCHEMBL24940877 0.80 CHRM5 (0.39) SIGMAR1ACHEOPRM1OPRK1OPRL1
SCHEMBL24921700 0.80 HRH1 (0.38) MEN1HTR4CYP2D6CYP3A4HRH3
SCHEMBL27267884 0.79 ACHE (0.37) HRH3SIGMAR1ACHEOPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed