SCHEMBL24920548

SCHEMBL24920548

COCc1ccnc(N2CCN(C)CC2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.48
AOC3 Q16853 1/20 0.45
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
HRH4 Q9H3N8 3/20 0.43
HTR3A P46098 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
HTR7 P34969 1/20 0.43
HTR6 P50406 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921040 0.88 AOC3 (0.44) ACHEAOC3CA12CA1CA2
SCHEMBL24921023 0.88 AOC3 (0.44) ACHEAOC3CA12CA1CA2
SCHEMBL24920520 0.86 MAPT (0.46) ACHEAOC3CA12CA1CA2
SCHEMBL24920536 0.85 ACHE (0.48) ACHEAOC3CA12CA1CA2
SCHEMBL24920523 0.84 ADRB1 (0.51) ACHEAOC3HRH4HTR3AHRH3
SCHEMBL30230267 0.83 HTR1A (0.56) ACHEHRH4HTR3AHTR1ADRD2
SCHEMBL16815333 0.81 ACHE (0.50) ACHEHRH4HTR3AHTR1ADRD2
SCHEMBL24920516 0.80 HSD17B10 (0.41) AOC3ALDH1A1CYP1A2HSD17B10
SCHEMBL24921022 0.79 AOC3 (0.38) ACHEAOC3HTR2A
SCHEMBL24921025 0.78 RXRA (0.39) AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed