SCHEMBL24934252

SCHEMBL24934252

CNC(=O)c1cccc(-c2ncco2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.49
PIP5K1C O60331 1/20 0.48
PIK3CA P42336 1/20 0.48
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
KDM5A P29375 1/20 0.47
KDM4C Q9H3R0 1/20 0.47
KDM5B Q9UGL1 1/20 0.47
GLRA3 O75311 1/20 0.46
GLRB P48167 1/20 0.46
MAP4K4 O95819 1/20 0.45
USP30 Q70CQ3 1/20 0.45
HPGDS O60760 1/20 0.44
FYN P06241 1/20 0.44
PLK1 P53350 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933996 0.86 ALDH1A1 (0.47) HDAC8GLRA3GLRBHPGDSALDH1A1
SCHEMBL30999881 0.86 ALDH1A1 (0.47) HDAC8GLRA3GLRBHPGDSALDH1A1
SCHEMBL9507238 0.84 BRD4 (0.48) CDK8GLRA3GLRBMAP4K4HPGDS
SCHEMBL31216543 0.83 KAT6A (0.44) HDAC8HDAC6GLRA3GLRBHPGDS
SCHEMBL6434655 0.83 GLRA3 (0.62) CDK8KDM4CGLRA3GLRBHPGDS
SCHEMBL17146451 0.83 GLRA3 (0.44) PIP5K1CPIK3CAGLRA3GLRBHPGDS
SCHEMBL939928 0.82 KEAP1 (0.55) HDAC6KDM5AKDM4CKDM5BGLRA3
SCHEMBL31558442 0.82 KEAP1 (0.55) HDAC6KDM5AKDM4CKDM5BGLRA3
SCHEMBL6433748 0.81 HPGDS (0.47) GLRA3GLRBHPGDSALDH1A1HPGD
SCHEMBL6573037 0.81 PRKCI (0.50) CDK8GLRA3GLRBUSP30HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023009475-A1 ROCK2 INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-02-02 WO disclosed