SCHEMBL2500368

SCHEMBL2500368

O=C(OC(=O)c1ccc(CBr)cc1)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.69
CES1 P23141 2/20 0.69
TDP1 Q9NUW8 2/20 0.48
KMT2A Q03164 2/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A3 Q01959 1/20 0.48
LMNA P02545 3/20 0.48
F2 P00734 1/20 0.48
TSHR P16473 3/20 0.48
ALDH1A1 P00352 3/20 0.48
TRPA1 O75762 1/20 0.48
PTPN1 P18031 1/20 0.45
GSK3B P49841 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.44
HIF1A Q16665 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2500365 0.92 CES2 (0.55) CES2CES1TDP1KMT2ASLC6A2
SCHEMBL8717537 0.83 LMNA (0.67) CES2CES1TDP1KMT2ASLC6A2
SCHEMBL775751 0.82 ALDH1A1 (0.61) CES2CES1TDP1KMT2ASLC6A2
SCHEMBL1352549 0.82 CES2 (1.00) CES2CES1LMNATSHRALDH1A1
SCHEMBL118227 0.82 CES2 (0.77) CES2CES1TDP1KMT2ALMNA
SCHEMBL4650584 0.81 KMT2A (0.76) CES2CES1TDP1KMT2ASLC6A2
SCHEMBL7616356 0.81 CES2 (0.59) CES2CES1TDP1KMT2AALDH1A1
SCHEMBL8983809 0.81 CES2 (0.59) CES2CES1TDP1KMT2ATSHR
SCHEMBL6777691 0.81 RAB9A (0.71) CES2CES1KMT2ALMNAALDH1A1
SCHEMBL52413 0.81 LMNA (0.70) CES2CES1TDP1KMT2ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8029979-B2 Method for determining the substrate specificity of an enzyme JPT PEPTIDE TECHNOLOGIES GMBH (DE) 2011-10-04 US disclosed
US-20060234308-A1 Method for determining the substrate specificity of an enzymatic activity and a device therefor JERINI AG (DE) 2006-10-19 US disclosed
US-20040171097-A1 Method for determining the substrate specificity of an enzymatic activity and a device therefor JERINI AG (DE) 2004-09-02 US disclosed