SCHEMBL250105

SCHEMBL250105

CN(C)C1(c2cccs2)CCC(N)CC1.N#CC(c1ccccc1)c1ccc(NC(=O)CCCC(=O)O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C1 Q04828 1/20 0.40
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 3/20 0.35
OPRL1 P41146 3/20 0.35
ENPP2 Q13822 4/20 0.35
POLB P06746 2/20 0.34
NAMPT P43490 1/20 0.34
MCHR1 Q99705 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249885 0.86 MAPT (0.43) ALDH1A1MAPTMEN1KMT2AENPP2
SCHEMBL251293 0.82 ENPP2 (0.42) ALDH1A1MAPTENPP2POLBTP53
SCHEMBL250636 0.82 LTA4H (0.52) ALDH1A1MAPTMEN1KMT2A
SCHEMBL4075171 0.77 ALDH1A1 (0.62) ALDH1A1AKR1C3AKR1C1MAPTMEN1
SCHEMBL4084421 0.77 OPRM1 (0.45) ALDH1A1MAPTOPRM1OPRL1MCHR1
SCHEMBL248430 0.76 THRB (0.37) ALDH1A1MAPTMEN1KMT2AOPRM1
SCHEMBL251283 0.75 OPRM1 (0.44) ALDH1A1OPRM1OPRL1
SCHEMBL4074080 0.75 OPRM1 (0.51) OPRM1OPRL1
SCHEMBL250033 0.75 OPRL1 (0.42) MAPTOPRM1OPRL1
SCHEMBL250470 0.75 OPRM1 (0.46) KMT2AOPRM1OPRL1ICMTALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US disclosed