SCHEMBL25019676

SCHEMBL25019676

CCOC(=O)c1c(CO)c2sc(C3=CC3C)nc2n1-c1nccs1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.34
CDC7 O00311 5/20 0.33
DBF4 Q9UBU7 5/20 0.33
ALDH1A1 P00352 4/20 0.33
PKM P14618 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
KDM4E B2RXH2 2/20 0.32
LMNA P02545 1/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
MAPT P10636 2/20 0.31
GAA P10253 1/20 0.31
ALOX15 P16050 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20745728 0.82 LMNA (0.41) MAPK1CDC7DBF4ALDH1A1PKM
SCHEMBL20745576 0.70 LMNA (0.41) MAPK1ALDH1A1PKMADORA2AADORA2B
SCHEMBL20746353 0.68 KDM4E (0.39) MAPK1ALDH1A1PKMKDM4ELMNA
SCHEMBL14549182 0.60 HDAC3 (0.54) ALDH1A1PKMNPC1RAB9A
SCHEMBL20028220 0.60 SMN1; SMN2 (0.49) ALDH1A1PKMKDM4ELMNAHPGD
SCHEMBL19975395 0.60 SCN9A (0.45) MAPK1ALDH1A1PKMADORA2AKDM4E
SCHEMBL13211356 0.59 HDAC3 (0.52) CDC7DBF4ALDH1A1PKMKDM4E
SCHEMBL9369759 0.58 NOTUM (0.52) MAPK1ALDH1A1PKMKDM4ELMNA
SCHEMBL837325 0.58 ALDH1A1 (0.55) MAPK1CDC7DBF4ALDH1A1PKM
SCHEMBL13174880 0.57 RAB9A (0.64) MAPK1ALDH1A1PKMMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3668512-B1 PYRUVATE KINASE MODULATORS AND USE THEREOF AGIOS PHARMACEUTICALS INC (US) 2023-02-15 EP disclosed