SCHEMBL25064044

SCHEMBL25064044

C=C(C)c1cc(F)c(Cl)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20076683 0.87 CYP3A4 (0.37)
SCHEMBL24931097 0.80 CES2 (0.50) CES2CES1
SCHEMBL16961740 0.80 CES2 (0.33) CES2CES1
SCHEMBL7910357 0.78 VRK1 (0.34) CES2CES1
SCHEMBL27417243 0.78 HDAC1 (0.48) CES2CES1
SCHEMBL23112583 0.76 CA5A (0.46) CES2CES1
SCHEMBL8296527 0.76 KCNQ3 (0.41) CES2CES1
SCHEMBL16954968 0.76
SCHEMBL14955991 0.75 HPGD (0.43)
SCHEMBL14956621 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12435054-B2 Therapeutic compounds and methods of use GENENTECH, INC. (US) 2025-10-07 US disclosed
EP-4185386-B1 HETEROCYCLIC INHIBITORS OF TEAD FOR TREATING CANCER GENENTECH INC (US) 2025-01-08 EP disclosed
US-20240208919-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2024-06-27 US disclosed
US-20240208919-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2024-06-27 US disclosed
US-11787775-B2 Therapeutic compounds and methods of use GENENTECH, INC. (US) 2023-10-17 US disclosed
US-11787775-B2 Therapeutic compounds and methods of use GENENTECH, INC. (US) 2023-10-17 US disclosed
US-11787775-B2 Therapeutic compounds and methods of use GENENTECH, INC. (US) 2023-10-17 US disclosed
CN-116234797-A Heterocyclic inhibitors of TEAD for the treatment of cancer 基因泰克公司 2023-06-06 CN disclosed
EP-4185386-A1 HETEROCYCLIC INHIBITORS OF TEAD FOR TREATING CANCER Genentech, Inc. (US) 2023-05-31 EP disclosed
US-20230054741-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-02-23 US disclosed
US-20230054741-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230054741-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE VHL, NQO1, PCSK9 CES2 152/4885CES1 706/4885
US-20240208919-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE VHL, NQO1, PCSK9 CES2 152/4885CES1 706/4885
US-11787775-B2 Therapeutic compounds and methods of use VHL, NQO1, PCSK9 CES2 152/4885CES1 706/4885
US-12435054-B2 Therapeutic compounds and methods of use VHL, NQO1, PCSK9 CES2 152/4885CES1 706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.