SCHEMBL25130855

SCHEMBL25130855

COc1nc(Cl)cc2c(Br)ccnc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 1/20 0.34
HIPK2 Q9H2X6 1/20 0.34
NSD2 O96028 2/20 0.33
CASP6 P55212 1/20 0.33
G6PD P11413 1/20 0.33
CCR4 P51679 1/20 0.33
APAF1 O14727 1/20 0.32
TDP2 O95551 1/20 0.32
CASP3 P42574 1/20 0.32
PPP1CA P62136 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
SAE1 Q9UBE0 1/20 0.32
UBA2 Q9UBT2 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27167385 0.83 CSNK2A1 (0.35) CSNK2A1HIPK2NSD2CASP6APAF1
SCHEMBL25130861 0.81 KDM4E (0.35) G6PDCCR4SMN1; SMN2KDM4EMEN1
SCHEMBL29923740 0.79 CSNK2A1 (0.33) CSNK2A1HIPK2NSD2CASP6APAF1
SCHEMBL24916320 0.79 CSNK2A1 (0.33) CSNK2A1HIPK2NSD2CASP6APAF1
SCHEMBL25130613 0.79 GRM4 (0.34) APAF1TDP2CASP3SENP8SENP7
SCHEMBL160724 0.74 NR1I3 (0.41) KDM4ETP53HSP90AA1PDCD1CD274
SCHEMBL20292984 0.73 NSD2 (0.40) NSD2CASP6G6PDAPAF1TDP2
SCHEMBL26639901 0.72 ALDH1A1 (0.43) CCR4SMN1; SMN2KDM4EMEN1KMT2A
SCHEMBL31729196 0.70 CCR4 (0.33) CSNK2A1HIPK2CCR4SMN1; SMN2KDM4E
SCHEMBL30657478 0.70 MEN1 (0.34) CCR4KDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023051628-A1 SOS1 INHIBITORS HAVING PYRIDO SIX-MEMBERED RING STRUCTURE 上海海和药物研究开发股份有限公司 2023-04-06 WO disclosed