SCHEMBL25149446

SCHEMBL25149446

COc1nc(C2CCC(C(F)(F)F)CC2)ccc1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.39
ROCK1 Q13464 1/20 0.39
TRPV3 Q8NET8 1/20 0.39
NNMT P40261 1/20 0.37
CDK8 P49336 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
GSK3B P49841 1/20 0.35
NR3C1 P04150 2/20 0.35
PGR P06401 2/20 0.35
NR3C2 P08235 2/20 0.35
AR P10275 2/20 0.35
PARP1 P09874 1/20 0.35
POLB P06746 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
TBK1 Q9UHD2 1/20 0.33
IRAK1 P51617 1/20 0.33
EGFR P00533 1/20 0.33
TEC P42680 1/20 0.33
BTK Q06187 1/20 0.33
PDCD1LG2 Q9BQ51 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30364759 0.87 TRPV3 (0.38) ROCK2TRPV3PARP1NR1H2NR1H3
SCHEMBL25149306 0.83 PARP15 (0.42) ROCK2ROCK1NNMTCDK8CDK19
SCHEMBL25148626 0.83 PARP15 (0.42) ROCK2ROCK1NNMTCDK8CDK19
SCHEMBL27906200 0.82 TRPV3 (0.39) ROCK2TRPV3PARP1POLBTBK1
SCHEMBL25149632 0.78 NNMT (0.41) ROCK2ROCK1NNMTGSK3BNR3C1
SCHEMBL30365013 0.76 LMNA (0.40) TRPV3POLB
SCHEMBL25148803 0.72 NR3C1 (0.40) ROCK2ROCK1NNMTGSK3BNR3C1
SCHEMBL3544818 0.71 NNMT (0.45) ROCK2ROCK1NNMTPOLBTDP1
SCHEMBL26618866 0.70 MAPK1 (0.41) NNMTPARP1POLBEGFRTEC
SCHEMBL28014566 0.70 NNMT (0.51) NNMTPARP1POLBTDP1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023062575-A1 CYCLIC VINYL SULFONE COMPOUNDS AS WRN INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-20 WO disclosed