SCHEMBL25149306

SCHEMBL25149306

COc1nc(C2CCCCC2)ccc1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 1/20 0.42
PARP10 Q53GL7 1/20 0.42
NR3C1 P04150 2/20 0.42
PGR P06401 2/20 0.42
NR3C2 P08235 2/20 0.42
AR P10275 2/20 0.42
CNR2 P34972 2/20 0.42
NNMT P40261 1/20 0.41
TACR3 P29371 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
PDE7A Q13946 1/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
GSK3B P49841 1/20 0.38
CDC7 O00311 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25148626 1.00 PARP15 (0.42) PARP15PARP10NR3C1PGRNR3C2
SCHEMBL25148734 0.86 PDCD1 (0.44) CNR2TACR3POLBTDP1KDM4E
SCHEMBL30364876 0.86 PDCD1 (0.44) CNR2TACR3POLBTDP1KDM4E
SCHEMBL25149632 0.83 NNMT (0.41) NR3C1PGRNR3C2ARNNMT
SCHEMBL25149446 0.83 ROCK2 (0.39) NR3C1PGRNR3C2ARNNMT
SCHEMBL25148803 0.82 NR3C1 (0.40) PARP15PARP10NR3C1PGRNR3C2
SCHEMBL4153908 0.81 NNMT (0.47) PARP15PARP10CNR2NNMTPDE7A
SCHEMBL30364997 0.73 LMNA (0.44) CNR2TACR3POLBMEN1MAPT
SCHEMBL21906150 0.73 PARP1 (0.38) PARP15PARP10CDC7KDM4EMEN1
SCHEMBL28014566 0.72 NNMT (0.51) NNMTPOLBTDP1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023062575-A1 CYCLIC VINYL SULFONE COMPOUNDS AS WRN INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-20 WO disclosed