SCHEMBL25218330

SCHEMBL25218330

OC(CC1CCN(CCc2ccccc2)CC1)c1cccnc1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
TSHR P16473 1/20 0.58
HTR2A P28223 1/20 0.58
HTR2C P28335 1/20 0.58
CCR3 P51677 1/20 0.51
HRH3 Q9Y5N1 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25253155 0.86 HTR2A (0.76) KDM4ECYP1A2CYP3A4CYP2D6TSHR
SCHEMBL4164304 0.83 KDM4E (0.55) KDM4ECYP1A2CYP3A4CYP2D6TSHR
Bromide SCHEMBL4173363 0.82 KDM4E (0.53) KDM4ECYP1A2CYP3A4CYP2D6TSHR
SCHEMBL4611120 0.78 KDM4E (0.49) KDM4ECYP1A2CYP3A4CYP2D6TSHR
SCHEMBL10350582 0.77 SIGMAR1 (0.54) CYP1A2CYP3A4CYP2D6TSHRCCR3
SCHEMBL10350000 0.76 SIGMAR1 (0.53) CYP1A2CYP3A4CYP2D6TSHRCCR3
SCHEMBL11631293 0.76 IDO1 (0.45) CYP1A2CYP3A4CYP2D6
Glemanserin SCHEMBL120012 0.74 HTR2A (1.00) KDM4ECYP1A2CYP3A4CYP2D6TSHR
SCHEMBL4611997 0.74 L3MBTL1 (0.53)
SCHEMBL4168265 0.74 SLC6A3 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023107547-A2 AZETIDINE AND SPIROAZETIDINE COMPOUNDS AND USES THEREOF Kineta, Inc. (US) 2023-06-15 WO disclosed
WO-2023107547-A2 AZETIDINE AND SPIROAZETIDINE COMPOUNDS AND USES THEREOF Kineta, Inc. (US) 2023-06-15 WO disclosed