SCHEMBL25222005

SCHEMBL25222005

COc1c(F)cc(F)c(I)c1F

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31
DBH P09172 1/20 0.30
TUBB1 Q9H4B7 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ACHE P22303 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25348552 0.83 TDP1 (0.33) CYP3A4MAPTPDGFRBPDGFRADBH
SCHEMBL22883762 0.83 TDP1 (0.36) CYP3A4MAPTPDGFRBPDGFRADBH
SCHEMBL3836660 0.83 ACHE (0.32) CYP3A4MAPTACHECYP19A1
SCHEMBL30407185 0.81 CA2 (0.42) CYP3A4MAPTTUBB1
SCHEMBL30977479 0.81 HSD17B10 (0.32) CYP3A4MAPT
SCHEMBL3841844 0.81 CA2 (0.42) CYP3A4MAPTTUBB1
SCHEMBL1224037 0.81 PTGS2 (0.35) CYP3A4MAPT
SCHEMBL23898583 0.81 HSD17B10 (0.32)
SCHEMBL31015911 0.81 PTGS2 (0.35) CYP3A4MAPT
SCHEMBL31015975 0.78 ILK (0.33) CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12466803-B2 BCKDK inhibitors and/or degraders PFIZER INC. (US) 2025-11-11 US disclosed
US-20230167080-A1 BCKDK INHIBITORS AND/OR DEGRADERS PFIZER INC. (US) 2023-06-01 US disclosed
US-20230167080-A1 BCKDK INHIBITORS AND/OR DEGRADERS PFIZER INC. (US) 2023-06-01 US disclosed
US-20230167080-A1 BCKDK INHIBITORS AND/OR DEGRADERS PFIZER INC. (US) 2023-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12466803-B2 BCKDK inhibitors and/or degraders BCKDK, KHK, PDK4 CYP3A4 720/4885MAPT 2447/4885PDGFRB 2338/4885
US-20230167080-A1 BCKDK INHIBITORS AND/OR DEGRADERS BCKDK, KHK, PDK4 CYP3A4 720/4885MAPT 2447/4885PDGFRB 2338/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.