SCHEMBL25259922

SCHEMBL25259922

COc1cnccc1[C@]1(O)C[C@H]2CC[C@@H](C1)N2C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
TSHR P16473 1/20 0.45
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP2C19 P33261 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
KDM4E B2RXH2 1/20 0.36
GRM5 P41594 2/20 0.36
HTR1A P08908 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25295383 1.00 ALDH1A1 (0.45) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL25436394 0.91 ALDH1A1 (0.41) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL25436389 0.91 ALDH1A1 (0.41) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL30020976 0.86 GPR119 (0.42) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL30325528 0.75 CCR2 (0.40) ALDH1A1MEN1KMT2AGAANPSR1
SCHEMBL30325596 0.73 CDK9 (0.45)
SCHEMBL24212057 0.71 GPR119 (0.35) ALDH1A1TSHRSMN1; SMN2DRD2DRD3
SCHEMBL2586854 0.71 GPR119 (0.42) MEN1KMT2AGAAHTTNPSR1
SCHEMBL17728500 0.69 TSHR (0.36) TSHRMEN1KMT2ASMN1; SMN2SLC6A2
SCHEMBL1267331 0.68 ALDH1A1 (0.55) ALDH1A1TSHRDRD2DRD3GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023136279-A1 CRYSTAL OF SUBSTITUTED PIPERIDINE COMPOUND, SALTS OF SUBSTITUTED PIPERIDINE COMPOUND, AND CRYSTALS THEREOF エーザイ・アール・アンド・ディー・マネジメント株式会社 2023-07-20 WO disclosed