SCHEMBL2527293

SCHEMBL2527293

CCCCCn1c2ncn(Br)c2c(=O)n2c(CCc3nc(Cc4cc(F)cc(F)c4)no3)nnc12

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.38
ADORA2A P29274 3/20 0.33
ALDH1A1 P00352 2/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
CNOT7 Q9UIV1 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2527362 0.88 ALDH1A1 (0.32) PPARGADORA2AALDH1A1PKMTSHR
SCHEMBL2527116 0.88 ADORA2A (0.38) ADORA2AALDH1A1SMN1; SMN2CNOT7
SCHEMBL2531387 0.87 ALDH1A1 (0.34) PPARGADORA2AALDH1A1SMN1; SMN2CNOT7
SCHEMBL2524833 0.87 PPARG (0.35) PPARGADORA2AALDH1A1PKMTSHR
SCHEMBL2523023 0.86 MAPT (0.38) PPARGADORA2AALDH1A1MAPK1SMN1; SMN2
SCHEMBL2527271 0.86 MEN1 (0.42) PPARGADORA2AALDH1A1SMN1; SMN2CNOT7
SCHEMBL2524932 0.85 HSP90AA1 (0.38) PPARGALDH1A1PKMMAPK1SMN1; SMN2
SCHEMBL2529251 0.85 PPARG (0.41) PPARGADORA2AALDH1A1SMN1; SMN2
SCHEMBL2528388 0.83 ALDH1A1 (0.35) ADORA2AALDH1A1SMN1; SMN2CNOT7
SCHEMBL2528328 0.82 TSHR (0.38) ADORA2AALDH1A1TSHRMAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039478-B2 Purinone derivatives as HM74A agonists INCYTE CORPORATION (US) 2011-10-18 US disclosed