SCHEMBL2528068

SCHEMBL2528068

CCCCCn1c2ncn(Br)c2c(=O)n2c(CCc3nc(C4(c5ccccc5)CC4)no3)nnc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ADORA2A P29274 6/20 0.36
CNOT7 Q9UIV1 4/20 0.35
TSHR P16473 3/20 0.32
NPSR1 Q6W5P4 2/20 0.32
HTT P42858 1/20 0.32
USP2 O75604 2/20 0.31
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
XBP1 P17861 1/20 0.31
RBP1 P09455 1/20 0.30
MEN1 O00255 1/20 0.30
LMNA P02545 1/20 0.30
GLA P06280 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2527366 0.85 ADORA2A (0.38) ALDH1A1SMN1; SMN2ADORA2APLK1APOBEC3G
SCHEMBL2527116 0.82 ADORA2A (0.38) ALDH1A1SMN1; SMN2ADORA2ACNOT7PDE4A
SCHEMBL561771 0.81 ADORA2A (0.38) ALDH1A1SMN1; SMN2ADORA2APLK1APOBEC3G
SCHEMBL2528328 0.79 TSHR (0.38) ALDH1A1SMN1; SMN2ADORA2ACNOT7TSHR
SCHEMBL2528388 0.78 ALDH1A1 (0.35) ALDH1A1SMN1; SMN2ADORA2ACNOT7
SCHEMBL2524833 0.78 PPARG (0.35) ALDH1A1SMN1; SMN2ADORA2ACNOT7TSHR
SCHEMBL2523023 0.77 MAPT (0.38) ALDH1A1SMN1; SMN2ADORA2ACNOT7HTT
SCHEMBL2527293 0.76 PPARG (0.38) ALDH1A1SMN1; SMN2ADORA2ACNOT7TSHR
SCHEMBL2531387 0.76 ALDH1A1 (0.34) ALDH1A1SMN1; SMN2ADORA2ACNOT7KDM4E
SCHEMBL2524932 0.76 HSP90AA1 (0.38) ALDH1A1SMN1; SMN2CNOT7HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039478-B2 Purinone derivatives as HM74A agonists INCYTE CORPORATION (US) 2011-10-18 US disclosed