SCHEMBL252888

SCHEMBL252888

Cc1ccc2cccnc2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
LMNA P02545 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP1A2 P05177 1/20 0.46
CCR1 P32246 4/20 0.46
CCR5 P51681 4/20 0.46
CCR8 P51685 3/20 0.46
GMNN O75496 1/20 0.46
TP53 P04637 1/20 0.46
HSP90AA1 P07900 1/20 0.46
MMP2 P08253 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
MMP9 P14780 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11992064 0.81 CCR1 (0.57) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL16125081 0.78 CYP1A2 (0.43) MEN1KMT2ACYP1A2CCR1CCR5
SCHEMBL9533951 0.77 ALDH1A1 (0.52) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL29354893 0.77 CCR1 (0.55) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL7509409 0.77 CCR1 (0.58) LMNAKDM4EKMT2ACYP1A2CCR1
SCHEMBL28304525 0.77 CCR1 (0.55) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL8193 0.77 CCR1 (0.55) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL1089189 0.76 ALDH1A1 (0.55) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL29400608 0.76 CCR1 (0.70) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL3193864 0.76 CCR1 (0.70) ALDH1A1LMNAKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 730 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240383856-A1 INHIBITORS OF TRANSGLUTAMINASES ZEDIRA GMBH (DE) 2024-11-21 US claimed
US-20240376055-A1 INHIBITORS OF TRANSGLUTAMINASES ZEDIRA GMBH (DE) 2024-11-14 US claimed
CN-118270777-A Application of nucleoside modified graphene oxide in chiral compound recognition 北京交通大学 2024-07-02 CN claimed
CN-110272417-B 2-methyl-1, 8-naphthyridine compound and preparation method and application thereof 五邑大学 2021-07-13 CN claimed
WO-2020253415-A1 2-METHYL-1,8-NAPHTHYRIDINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREFOR 五邑大学 2020-12-24 WO claimed
CN-110272417-A 2- methyl-1,8- naphthyridine type compound and the preparation method and application thereof 五邑大学 2019-09-24 CN claimed
CN-106045996-B A kind of 2- (2 '-hydroxy styrenes base) naphthyridines probe reagents and its preparation and application 贵州大学 2018-06-19 CN claimed
CN-104974181-B 1, 8-naphthyridine binuclear copper (I) complex, preparation method and application 中国科学院理化技术研究所 2017-01-25 CN claimed
CN-106252686-A A kind of can the hydrogen energy power generation system of hydrogen-preparing hydrogen-storing 温州集智科技有限公司 2016-12-21 CN claimed
CN-106045996-A 2-(2'-hydroxyl styryl) naphthyridine probe reagent and preparation and application thereof 贵州大学 2016-10-26 CN claimed
EP-4159727-B1 INHIBITORS OF (ALPHA-V)(BETA-6) INTEGRIN MORPHIC THERAPEUTIC INC (US) 2026-04-08 EP disclosed
EP-4665458-A1 INHIBITING ALPHA V BETA8 INTEGRIN Morphic Therapeutic, Inc. (US) 2025-12-24 EP disclosed
US-12459942-B2 Inhibiting (α-v)(β-6) integrin MORPHIC THERAPEUTIC, INC. (US) 2025-11-04 US disclosed
US-12415796-B2 Inhibitors of (αv)(β6) integrin MORPHIC THERAPEUTIC, INC. (US) 2025-09-16 US disclosed
WO-2025149628-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF NICOTINAMIDE N-METHYL TRANSFERASE ASTRAZENECA AB (SE) 2025-07-17 WO disclosed
US-4273862-A ANIONIC CYANINE DYE, HYDROQUINONE FRBRLOPRT MITSUBISHI PAPER MILLS, LTD. (JP) 1981-06-16 US disclosed
US-4259439-A DIMETHINECYANINE DYE SENSITIZER MITSUBISHI PAPER MILLS, LTD. (JP) 1981-03-31 US disclosed
US-4175965-A SILVER HALIDE EMULSION CONTAINING AN ELECTRON ACCEPTOR AND A SENSITIZING DYE MITSUBISHI PAPER MILLS, LTD. (JP) 1979-11-27 US disclosed
US-4147554-A 5,6-DIHYDRO-PYRROLO(2,1-A)ISOQUINOLINES MITSUBISHI PAPER MILLS, LTD. (JP) 1979-04-03 US disclosed
US-4134769-A BETAINE AND ANIONIC TYPE CYANINE DYES MITSUBISHI PAPER MILLS, LTD. (JP) 1979-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12459942-B2 Inhibiting (α-v)(β-6) integrin ITGB6, ITGA6, ITGAV ALDH1A1 1629/4885LMNA 2251/4885KDM4E 3386/4885
US-12415796-B2 Inhibitors of (αv)(β6) integrin ITGB6, ITGA6, ITGAV ALDH1A1 2417/4885LMNA 2741/4885KDM4E 3739/4885
US-20240383856-A1 INHIBITORS OF TRANSGLUTAMINASES TGM2, TGM3, TGM1 ALDH1A1 1825/4885LMNA 2598/4885KDM4E 967/4885
US-20240376055-A1 INHIBITORS OF TRANSGLUTAMINASES TGM2, TGM3, TGM1 ALDH1A1 1825/4885LMNA 2598/4885KDM4E 967/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.