SCHEMBL25307353

SCHEMBL25307353

CC(C)(C)OC(=O)N1CC2(CCC2)CC(O)(c2c[nH]c3ncccc23)C1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.38
HSD11B1 P28845 8/20 0.38
MAP2K1 Q02750 1/20 0.37
POLB P06746 1/20 0.37
KIT P10721 1/20 0.37
DTYMK P23919 1/20 0.36
JAK3 P52333 2/20 0.35
CCNK O75909 1/20 0.35
CDK12 Q9NYV4 1/20 0.35
MET P08581 1/20 0.35
AXL P30530 1/20 0.35
NAMPT P43490 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25426035 0.96 CYP11B2 (0.39) CYP11B2HSD11B1MAP2K1POLBKIT
SCHEMBL30509709 0.96 CYP11B2 (0.39) CYP11B2HSD11B1MAP2K1POLBKIT
SCHEMBL30509700 0.86 HSD11B1 (0.42) CYP11B2HSD11B1MAP2K1POLBDTYMK
SCHEMBL25429671 0.86 HSD11B1 (0.42) CYP11B2HSD11B1MAP2K1POLBDTYMK
SCHEMBL25427796 0.79 HSD11B1 (0.41) HSD11B1MAP2K1POLBDTYMKJAK3
SCHEMBL30509712 0.79 HSD11B1 (0.41) HSD11B1MAP2K1POLBDTYMKJAK3
SCHEMBL30509683 0.78 HSD11B1 (0.42) HSD11B1MAP2K1POLBDTYMKJAK3
SCHEMBL25428242 0.78 HSD11B1 (0.42) HSD11B1MAP2K1POLBDTYMKJAK3
SCHEMBL25866544 0.78 MAP2K1 (0.39) HSD11B1MAP2K1POLBDTYMKJAK3
SCHEMBL1815353 0.74 HSD11B1 (0.61) HSD11B1MAP2K1POLBDTYMKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4466266-B1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS TRANSNEURAL THERAPEUTICS INC (US) 2026-04-08 EP disclosed
US-12486268-B2 Fused heterocycles as 5-HT2A receptor agonists Transneural Therapeutics, Inc. (US) 2025-12-02 US disclosed
US-12459944-B2 Fused heterocycles as 5-HT2A receptor agonists Transneural Therapeutics, Inc. (US) 2025-11-04 US disclosed
US-20250243199-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. (US) 2025-07-31 US disclosed
US-20240425503-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. 2024-12-26 US disclosed
EP-4466266-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. (US) 2024-11-27 EP disclosed
WO-2023141225-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS ONSERO THERAPEUTICS INC. (US) 2023-07-27 WO disclosed
WO-2023141225-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS ONSERO THERAPEUTICS INC. (US) 2023-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12459944-B2 Fused heterocycles as 5-HT2A receptor agonists HTR2A, HTR2C, HTR5A CYP11B2 486/4885HSD11B1 2233/4885MAP2K1 2999/4885
US-20250243199-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS HTR2A, HTR2C, HTR5A CYP11B2 486/4885HSD11B1 2233/4885MAP2K1 2999/4885
US-20240425503-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS HTR2A, HTR2C, HTR1A CYP11B2 616/4885HSD11B1 2614/4885MAP2K1 3311/4885
US-12486268-B2 Fused heterocycles as 5-HT2A receptor agonists HTR2A, HTR2C, HTR5A CYP11B2 486/4885HSD11B1 2233/4885MAP2K1 2999/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.