Bromide

Bromide

SCHEMBL2531329

Br.Ic1ccc(CN2C=CN(Cc3ccc(I)cc3)C2)cc1

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 1/20 0.33
HIF1A Q16665 2/20 0.36
EPAS1 Q99814 2/20 0.36
CYP3A4 P08684 2/20 0.35
IDO1 P14902 2/20 0.35
APP P05067 2/20 0.34
HTR2C P28335 1/20 0.33
FAAH O00519 1/20 0.33
HRH3 Q9Y5N1 2/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12220165 0.98 CYP3A4 (0.37) HIF1AEPAS1CYP3A4IDO1APP
Bromide SCHEMBL28054765 0.87 SIGMAR1 (0.34) HIF1AEPAS1CYP3A4IDO1HTR2C
SCHEMBL28331223 0.84 SIGMAR1 (0.35) HIF1AEPAS1CYP3A4IDO1APP
Hydrochloric Acid SCHEMBL28925128 0.83 SIGMAR1 (0.34) HIF1AEPAS1CYP3A4IDO1HTR2C
SCHEMBL28518181 0.79 SIGMAR1 (0.32) HIF1AEPAS1SIGMAR1HTR2A
Bromide SCHEMBL2529296 0.78 RAB9A (0.43) IDO1
Bromide SCHEMBL2530199 0.78 KDM4E (0.46) IDO1HTR2A
Bromide SCHEMBL1046639 0.77 SIGMAR1 (0.50) SIGMAR1
Hydrochloric Acid SCHEMBL2533088 0.76 ALDH1A1 (0.47) IDO1SIGMAR1
SCHEMBL12220123 0.76 KDM4E (0.47) IDO1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8632914-B2 Triazolium and imidazolium salts and uses thereof UNIVERSITY HEALTH NETWORK (CA) 2014-01-21 US disclosed
US-20110257235-A1 TRIAZOLIUM AND IMIDAZOLIUM SALTS AND USES THEREOF UNIVERSITY HEALTH NETWORK (CA) 2011-10-20 US disclosed
WO-2010025558-A1 TRIAZOLIUM AND IMIDAZOLIUM SALTS AND USES THEREOF AS ANTIMALARIALS UNIVERSITY HAEALTH NETWORK (CA) 2010-03-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110257235-A1 TRIAZOLIUM AND IMIDAZOLIUM SALTS AND USES THEREOF ARG2, ARG1, CIT SIGMAR1 209/4885HIF1A 4122/4885EPAS1 4836/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.