Benzimidazole

Benzimidazole

SCHEMBL2540653

CCN.c1ccc2[nH]cnc2c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.46
KDM4E B2RXH2 5/20 0.44
MAPT P10636 2/20 0.44
RAD52 P43351 1/20 0.44
MMP12 P39900 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
PDPK1 O15530 1/20 0.41
CA12 O43570 1/20 0.41
PARP1 P09874 1/20 0.41
ALOX15 P16050 1/20 0.41
CA9 Q16790 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
ALDH1A1 P00352 4/20 0.40
HPGD P15428 3/20 0.40
QPCT Q16769 3/20 0.40
RAB9A P51151 2/20 0.40
HTT P42858 1/20 0.40
QPCTL Q9NXS2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzimidazole SCHEMBL3540518 0.98 KDM4E (0.47) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL8010735 0.92 MMP12 (0.44) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL3181865 0.92 MMP12 (0.44) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL29285060 0.90 MMP12 (0.43) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL5317931 0.88 CTNNB1 (0.44) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL5404384 0.87 PRKCI (0.52) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL29218507 0.87 MMP12 (0.47) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL6009 0.87
Benzimidazole SCHEMBL461969 0.87 SMN1; SMN2 (0.50) PRKCIKDM4EMAPTRAD52MMP12
Benzimidazole SCHEMBL29358377 0.87

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114149419-A Oxadiazole drug molecule for medical nursing sterilization and disinfection and preparation method and application thereof 河南科技大学第一附属医院 2022-03-08 CN claimed
CN-114149419-A Oxadiazole drug molecule for medical nursing sterilization and disinfection and preparation method and application thereof 河南科技大学第一附属医院 2022-03-08 CN disclosed
EP-2560953-B1 INHIBITORS OF GLUTAMINYL CYCLASE PROBIODRUG AG (DE) 2016-01-06 EP disclosed
US-8541596-B2 Inhibitors PROBIODRUG AG (DE) 2013-09-24 US disclosed
EP-2560953-A2 NOVEL INHIBITORS Probiodrug AG (DE) 2013-02-27 EP disclosed
WO-2011131748-A2 NOVEL INHIBITORS PROBIODRUG AG (DE) 2011-10-27 WO disclosed
US-20110262388-A1 NOVEL INHIBITORS PROBIODRUG AG (DE) 2011-10-27 US disclosed
US-7705031-B2 Benzimidazoles useful as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-04-27 US disclosed
US-20080306129-A1 BENZIMIDAZOLES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED 2008-12-11 US disclosed
US-7309716-B2 Benzimidazoles useful as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-12-18 US disclosed
CN-1902181-A Benzimidazoles useful as modulators of ion channels VERTEX PHARMA (US) 2007-01-24 CN disclosed
US-20050209282-A1 Benzimidazoles useful as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED 2005-09-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209282-A1 Benzimidazoles useful as modulators of ion channels KCNJ11, KCNJ1, KCNJ2 PRKCI 1004/4885KDM4E 1468/4885MAPT 4227/4885
US-20110262388-A1 NOVEL INHIBITORS GLUL, QPCT, GLS PRKCI 1823/4885KDM4E 693/4885MAPT 3971/4885
US-20080306129-A1 BENZIMIDAZOLES USEFUL AS MODULATORS OF ION CHANNELS KCNJ11, KCNJ1, KCNJ2 PRKCI 1004/4885KDM4E 1468/4885MAPT 4227/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.