SCHEMBL25453078

SCHEMBL25453078

Cc1cc(Nc2ccccn2)ccc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.50
ALDH1A1 P00352 2/20 0.50
THRB P10828 1/20 0.50
ALOX15 P16050 1/20 0.50
RECQL P46063 1/20 0.50
HIF1A Q16665 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
RAB9A P51151 4/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MEN1 O00255 1/20 0.46
MAPK10 P53779 1/20 0.46
GFER P55789 1/20 0.46
KMT2A Q03164 1/20 0.46
KDR P35968 1/20 0.43
NPC1 O15118 3/20 0.41
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30502777 1.00 CYP3A4 (0.50) CYP3A4ALDH1A1THRBALOX15RECQL
SCHEMBL25175479 0.85 RAB9A (0.63) CYP3A4ALDH1A1RAB9ANPSR1MEN1
SCHEMBL25453077 0.81 MEN1 (0.48) RAB9AMEN1MAPK10GFERKMT2A
SCHEMBL30502751 0.81 MEN1 (0.48) RAB9AMEN1MAPK10GFERKMT2A
SCHEMBL2309841 0.81 RAB9A (0.48) CYP3A4ALDH1A1RAB9ANPSR1MEN1
SCHEMBL23609451 0.77 ALDH1A1 (0.50) CYP3A4ALDH1A1THRBALOX15RECQL
SCHEMBL29973206 0.77 ALDH1A1 (0.50) CYP3A4ALDH1A1THRBALOX15RECQL
SCHEMBL3040658 0.77 KDR (0.52) ALDH1A1ALOX15TDP1RAB9ANPSR1
SCHEMBL11511767 0.76 CYP3A4 (0.77) CYP3A4ALDH1A1THRBALOX15RECQL
SCHEMBL2127369 0.75 ALDH1A1 (0.70) CYP3A4ALDH1A1THRBALOX15RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081800-A1 ALPHA-2A ADRENERGIC RECEPTOR MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-05-11 WO disclosed