SCHEMBL2546401

SCHEMBL2546401

O=C1C2CCCCC2C(=O)N1CC1CCCCC1CN1CCN(c2cc3ccccc3cn2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.46
KCNH2 Q12809 3/20 0.44
DRD2 P14416 4/20 0.43
HTR2A P28223 4/20 0.43
HTR1A P08908 4/20 0.43
DRD3 P35462 4/20 0.43
HTR2C P28335 3/20 0.43
ADRA2C P18825 2/20 0.43
HTR2B P41595 2/20 0.43
CHRM2 P08172 2/20 0.43
ADRA2A P08913 2/20 0.43
DRD1 P21728 2/20 0.43
TBXA2R P21731 2/20 0.43
SLC6A2 P23975 2/20 0.43
ADRA1A P35348 2/20 0.43
SLC6A3 Q01959 2/20 0.43
ABCB11 O95342 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADRA2B P18089 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2541954 0.88 DRD2 (0.58) HTR3AKCNH2DRD2HTR2AHTR1A
SCHEMBL2544767 0.83 DRD2 (0.57) KCNH2DRD2HTR2AHTR1ADRD3
SCHEMBL2539519 0.77 DRD2 (0.50) KCNH2DRD2HTR2AHTR1ADRD3
SCHEMBL2541214 0.77 HTR1A (0.52) KCNH2DRD2HTR2AHTR1ADRD3
SCHEMBL2543290 0.76 HTR2A (0.52) KCNH2DRD2HTR2AHTR1ADRD3
SCHEMBL2546369 0.73 DRD2 (0.57) KCNH2DRD2HTR2AHTR1AHTR7
SCHEMBL2540314 0.73 DRD2 (0.63) KCNH2DRD2HTR2AHTR1ADRD3
SCHEMBL2544371 0.72 RAB9A (0.67) DRD2HTR2AHTR1ADRD3HTR2C
SCHEMBL2538137 0.72
SCHEMBL2547414 0.72 DRD2 (0.79) KCNH2DRD2HTR2AHTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563790-B1 A PROCESS OF A QUATERNARY AMMONIUM SALT SUMITOMO DAINIPPON PHARMA CO LTD (JP) 2016-09-14 EP disclosed
US-9309255-B2 Process of a quaternary ammonium salt SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2016-04-12 US disclosed
US-20150087830-A1 PROCESS OF A QUATERNARY AMMONIUM SALT SUMITOMO DAINIPPON PHARMA CO., LTD 2015-03-26 US disclosed
US-8921551-B2 Process of a quaternary ammonium salt SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2014-12-30 US disclosed
US-20140256939-A1 PROCESS OF PREPARING A QUATERNARY AMMONIUM SALT USING PHOSPHATE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2014-09-11 US disclosed
US-20140031548-A1 PROCESS OF A QUATERNARY AMMONIUM SALT USING PHOSPHATE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2014-01-30 US disclosed
US-8586737-B2 Process of a quaternary ammonium salt using phosphate DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2013-11-19 US disclosed
US-20110263847-A1 PROCESS OF A QUATERNARY AMMONIUM SALT DAINIPPON SUMITOMO PHARMA CO, LTD. (JP) 2011-10-27 US disclosed
US-20110263848-A1 PROCESS OF A QUATERNARY AMMONIUM SALT USING PHOSPHATE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150087830-A1 PROCESS OF A QUATERNARY AMMONIUM SALT KAT5, ATP1B2, QARS1 HTR3A 4562/4885KCNH2 132/4885DRD2 3458/4885
US-20140031548-A1 PROCESS OF A QUATERNARY AMMONIUM SALT USING PHOSPHATE PHPT1, SLC34A2, SLC34A3 HTR3A 4687/4885KCNH2 383/4885DRD2 4460/4885
US-20110263847-A1 PROCESS OF A QUATERNARY AMMONIUM SALT KAT5, ATP1B2, QARS1 HTR3A 4562/4885KCNH2 132/4885DRD2 3458/4885
US-20110263848-A1 PROCESS OF A QUATERNARY AMMONIUM SALT USING PHOSPHATE PHPT1, SLC34A2, SLC34A3 HTR3A 4687/4885KCNH2 383/4885DRD2 4460/4885
US-20140256939-A1 PROCESS OF PREPARING A QUATERNARY AMMONIUM SALT USING PHOSPHATE AGPS, SLC34A3, SLC34A1 HTR3A 4648/4885KCNH2 248/4885DRD2 4238/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.