SCHEMBL2548181

SCHEMBL2548181

O=S(=O)(CC1CCN(CC2CC2)C1)c1ccc(CNC2CCCC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.43
POLB P06746 2/20 0.41
ACHE P22303 8/20 0.41
BACE1 P56817 8/20 0.41
BCHE P06276 6/20 0.41
FABP6 P51161 1/20 0.40
HDAC1 Q13547 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2551564 0.83 HRH3 (0.45) HRH3POLBACHEBACE1BCHE
SCHEMBL2554540 0.83 KDM4E (0.47) HRH3POLBACHEBACE1BCHE
SCHEMBL2555072 0.70 KCNH2 (0.49) HRH3POLBFABP6MEN1KMT2A
SCHEMBL2555109 0.70 KDM4E (0.48) HRH3POLBACHEBACE1BCHE
SCHEMBL2547933 0.70 KDM4E (0.48) HRH3POLBACHEBACE1BCHE
SCHEMBL7716908 0.70 KDM4E (0.48) HRH3POLBACHEBACE1BCHE
SCHEMBL4940261 0.69 HRH3 (0.58) HRH3POLBHDAC1
SCHEMBL7716923 0.69 SMN1; SMN2 (0.54) HRH3POLBFABP6MEN1KMT2A
SCHEMBL7356760 0.69 DRD2 (0.56)
SCHEMBL20492777 0.69 ACHE (0.68) ACHEBACE1BCHEFABP6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed