SCHEMBL2548635

SCHEMBL2548635

CN1CCN(CCCN2c3c[c]ccc3Sc3ccccc32)CC1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 11/20 0.78
LMNA P02545 4/20 0.64
MAPT P10636 4/20 0.64
MAPK1 P28482 4/20 0.64
SMN1; SMN2 Q16637 4/20 0.64
HTR1A P08908 4/20 0.64
ADRA2A P08913 4/20 0.64
CHRM1 P11229 4/20 0.64
DRD2 P14416 4/20 0.64
ADRA2C P18825 4/20 0.64
DRD1 P21728 4/20 0.64
SLC6A2 P23975 4/20 0.64
HTR2A P28223 4/20 0.64
SLC6A4 P31645 4/20 0.64
ADRA1A P35348 4/20 0.64
HRH1 P35367 4/20 0.64
DRD3 P35462 4/20 0.64
SLC6A3 Q01959 4/20 0.64
KCNH2 Q12809 4/20 0.64
TP53 P04637 3/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Perazine SCHEMBL29390464 0.88 KDM1A (1.00) KDM1ALMNAMAPTMAPK1SMN1; SMN2
Perazine SCHEMBL147165 0.88 KDM1A (1.00) KDM1ALMNAMAPTMAPK1SMN1; SMN2
Perazine SCHEMBL6644457 0.87 KDM1A (0.97) KDM1ALMNAMAPTMAPK1SMN1; SMN2
Perazine SCHEMBL2237726 0.87 KDM1A (0.97) KDM1ALMNAMAPTMAPK1SMN1; SMN2
SCHEMBL6859184 0.86 KDM1A (0.94) KDM1ALMNAMAPTMAPK1SMN1; SMN2
Perazine SCHEMBL10531680 0.81 KDM1A (0.84) KDM1ALMNAMAPTMAPK1SMN1; SMN2
SCHEMBL4399786 0.81 KDM1A (0.70) KDM1ALMNAMAPTMAPK1SMN1; SMN2
SCHEMBL10973127 0.81 KDM1A (0.84) KDM1ALMNAMAPTMAPK1SMN1; SMN2
SCHEMBL2615404 0.79 KDM1A (0.80) KDM1ALMNAMAPTMAPK1SMN1; SMN2
SCHEMBL12083350 0.79 FPR2 (0.89) KDM1ALMNAMAPTMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552323-A1 COMBINATION THERAPY Follica, Inc. (US) 2013-02-06 EP disclosed
WO-2011123218-A1 COMBINATION THERAPY FOLLICA, INC. (US) 2011-10-06 WO disclosed
WO-2007041463-A2 ELECTRICAL DEVICES AND ANTI-SCARRING DRUG COMBINATIONS COMBINATORX, INCORPORATED (US) 2007-04-12 WO disclosed