SCHEMBL2550157

SCHEMBL2550157

C=CCOc1cccc2c1Cc1ccccc1-2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.54
ADRA2B P18089 2/20 0.54
ADRA2C P18825 2/20 0.54
PNMT P11086 1/20 0.45
HTR1A P08908 2/20 0.43
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
LIG1 P18858 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
MAPT P10636 2/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2A6 P11509 1/20 0.38
PTPRC P08575 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15938601 0.92 ADRA2A (0.49) ADRA2AADRA2BADRA2CPNMTHTR1A
SCHEMBL895389 0.84 CTSS (0.46) ADRA2AADRA2BADRA2CPNMTHPGD
SCHEMBL3789485 0.81 PNMT (0.42) ADRA2AADRA2BADRA2CPNMTTSHR
SCHEMBL15938603 0.80 ADRA2A (0.39) ADRA2AADRA2BADRA2CPNMTHTR1A
SCHEMBL21951946 0.80 PNMT (0.50) PNMTHPGDKDM4EALDH1A1MAPT
SCHEMBL23501513 0.80 MAPT (0.41) ADRA2AADRA2BADRA2CPNMTMAPK1
SCHEMBL28066660 0.79 PNMT (0.49) PNMTALDH1A1MAPTPTPRCL3MBTL1
SCHEMBL14803713 0.79 PNMT (0.45) PNMTHPGDMAPK1KDM4EALDH1A1
SCHEMBL3807830 0.77 MAOA (0.46) ADRA2AADRA2BADRA2CHTR1AHPGD
SCHEMBL15141606 0.76 PNMT (0.49) PNMTHPGDMAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130090031-A1 COMPOSITE FILM MATERIAL COMPRISING A RESIN OF FLUORENE CROTONATE, FLUORENE CINNAMATE, FLUORENE ACRYLATE, FLUORENE METHACRYLATE, FLUORENE ALLYLETHER OR A COMBINATION THEREOF FERRANIA TECHNOLOGIES S.P.A. (IT) 2013-04-11 US disclosed
EP-2556113-A1 COMPOSITE FILM MATERIAL COMPRISING A RESIN OF FLUORENE CROTONATE, FLUORENE CINNAMATE, FLUORENE ACRYLATE, FLUORENE METHACRYLATE, FLUORENE ALLYLETHER OR A COMBINATION THEREOF Ferrania Technologies S.p.A. (IT) 2013-02-13 EP disclosed
EP-2556113-A1 COMPOSITE FILM MATERIAL COMPRISING A RESIN OF FLUORENE CROTONATE, FLUORENE CINNAMATE, FLUORENE ACRYLATE, FLUORENE METHACRYLATE, FLUORENE ALLYLETHER OR A COMBINATION THEREOF Ferrania Technologies S.p.A. (IT) 2013-02-13 EP disclosed
WO-2011124522-A1 COMPOSITE FILM MATERIAL COMPRISING A RESIN OF FLUORENE CROTONATE, FLUORENE CINNAMATE, FLUORENE ACRYLATE, FLUORENE METHACRYLATE, FLUORENE ALLYLETHER OR A COMBINATION THEREOF FERRANIA TECHNOLOGIES S.P.A. (IT) 2011-10-13 WO disclosed
WO-2011124522-A1 COMPOSITE FILM MATERIAL COMPRISING A RESIN OF FLUORENE CROTONATE, FLUORENE CINNAMATE, FLUORENE ACRYLATE, FLUORENE METHACRYLATE, FLUORENE ALLYLETHER OR A COMBINATION THEREOF FERRANIA TECHNOLOGIES S.P.A. (IT) 2011-10-13 WO disclosed