SCHEMBL25501974

SCHEMBL25501974

Nc1nc(Cl)c(I)cc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
CYP3A4 P08684 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.37
TSHR P16473 1/20 0.37
CASP1 P29466 1/20 0.37
SLC9A1 P19634 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CISD1 Q9NZ45 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1301224 0.82 KEAP1 (0.60) KEAP1NFE2L2SMN1; SMN2TSHRCASP1
SCHEMBL23674282 0.82 IDO1 (0.38) CYP3A4CASP1SLC9A1ALDH1A1TDP1
SCHEMBL29795353 0.81 SLC9A1 (0.46) KEAP1NFE2L2CYP3A4SMN1; SMN2TSHR
SCHEMBL22666874 0.81 SLC9A1 (0.46) KEAP1NFE2L2CYP3A4SMN1; SMN2TSHR
SCHEMBL20298359 0.78 ALDH1A1 (0.46) KEAP1NFE2L2CYP3A4SMN1; SMN2SLC9A1
SCHEMBL24659358 0.78 KEAP1 (0.42) KEAP1NFE2L2CYP3A4SMN1; SMN2SLC9A1
SCHEMBL23674344 0.75 SLC9A1 (0.61) KEAP1NFE2L2CYP3A4SMN1; SMN2TSHR
SCHEMBL443877 0.73 KHK (0.35) TDP1
SCHEMBL4736844 0.73 CA12 (0.46) KEAP1CYP3A4SMN1; SMN2TSHRCASP1
SCHEMBL1317569 0.73 ALDH1A1 (0.41) KEAP1NFE2L2CYP3A4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023088291-A1 AROMATIC AMINE COMPOUND AND APPLICATION THEREOF 武汉众诚康健生物医药科技有限公司 2023-05-25 WO disclosed