SCHEMBL29795353

SCHEMBL29795353

Nc1nc(Cl)c(Cl)cc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.46
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
CYP3A4 P08684 1/20 0.41
ALDH1A1 P00352 5/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TSHR P16473 2/20 0.39
TP53 P04637 1/20 0.39
CASP1 P29466 1/20 0.39
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
POLB P06746 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22666874 1.00 SLC9A1 (0.46) SLC9A1KEAP1NFE2L2CYP3A4ALDH1A1
SCHEMBL23674344 0.86 SLC9A1 (0.61) SLC9A1KEAP1NFE2L2CYP3A4ALDH1A1
SCHEMBL24755247 0.84 SLC9A1 (0.50) SLC9A1ALDH1A1CASP1POLBKDM4E
SCHEMBL7540414 0.82 KEAP1 (0.46) KEAP1NFE2L2ALDH1A1SMN1; SMN2TSHR
SCHEMBL29406550 0.81 KEAP1 (0.64) KEAP1NFE2L2ALDH1A1SMN1; SMN2TSHR
SCHEMBL2566963 0.81 KEAP1 (0.64) KEAP1NFE2L2ALDH1A1SMN1; SMN2TSHR
SCHEMBL24659358 0.81 KEAP1 (0.42) SLC9A1KEAP1NFE2L2CYP3A4ALDH1A1
SCHEMBL20298359 0.81 ALDH1A1 (0.46) SLC9A1KEAP1NFE2L2CYP3A4ALDH1A1
SCHEMBL25501974 0.81 KEAP1 (0.42) SLC9A1KEAP1NFE2L2CYP3A4ALDH1A1
SCHEMBL20296487 0.81 SLC9A1 (0.44) SLC9A1KEAP1NFE2L2CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022262686-A1 KRAS G12D INHIBITORS JINGRUI BIOPHARMA CO., LTD. (CN) 2022-12-22 WO disclosed
WO-2022171191-A1 COMPOUNDS AS ANTICANCER AGENTS JINGRUI BIOPHARMA CO., LTD. (CN) 2022-08-18 WO disclosed