SCHEMBL25532

SCHEMBL25532

Nc1ccc(S(=O)(=O)N2CC2)c2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
ALDH1A1 P00352 5/20 0.55
TSHR P16473 5/20 0.55
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
NPC1 O15118 1/20 0.49
ATM Q13315 1/20 0.49
HTT P42858 2/20 0.48
LMNA P02545 2/20 0.48
MCOLN3 Q8TDD5 1/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TTR P02766 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104945 0.89 CYP3A4 (0.57) POLBSMN1; SMN2ALDH1A1TSHRKMT2A
SCHEMBL7837749 0.81 SMN1; SMN2 (0.77) SMN1; SMN2ALDH1A1TSHRKMT2AMEN1
SCHEMBL13788913 0.79 KMT2A (0.63) POLBSMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL4449287 0.77 TTR (0.51) POLBSMN1; SMN2KMT2AMEN1ATM
Hydrochloric Acid SCHEMBL4448322 0.76 TTR (0.50) POLBSMN1; SMN2KMT2AMEN1ATM
SCHEMBL108422 0.75 LDHA (0.64) ALDH1A1TSHRCYP3A4CYP2C9HPGD
SCHEMBL4455037 0.75 KMT2A (0.60) POLBSMN1; SMN2TSHRKMT2AMEN1
SCHEMBL8564336 0.74 MEN1 (0.83) SMN1; SMN2ALDH1A1TSHRKMT2AMEN1
SCHEMBL8842866 0.74 KDM4E (0.57) POLBALDH1A1TSHRHTTKDM4E
Hydrochloric Acid SCHEMBL4452980 0.74 KMT2A (0.59) POLBSMN1; SMN2TSHRKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 268 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12203936-B2 Detection of glutathionylated proteins UNIVERSITEIT MAASTRICHT (NL) 2025-01-21 US claimed
US-11927593-B2 High-throughput single molecule protein identification THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2024-03-12 US claimed
US-20210311057-A1 DETECTION OF GLUTATHIONYLATED PROTEINS THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2021-10-07 US claimed
US-20200271661-A1 HIGH-THROUGHPUT SINGLE MOLECULE PROTEIN IDENTIFICATION THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2020-08-27 US claimed
US-10466248-B2 High-throughput single molecule protein identification THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2019-11-05 US claimed
US-20180224452-A1 DETECTION OF GLUTATHIONYLATED PROTEINS THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2018-08-09 US claimed
CN-108051584-A Development and application of non-bilirubin-bound fluorescent probe 阿兰·马克·克莱费尔德 2018-05-18 CN claimed
CN-104220877-B Development and application of non-bilirubin-bound fluorescent probe 阿兰·马克·克莱费尔德 2018-05-15 CN claimed
US-20160238612-A1 HIGH-THROUGHPUT SINGLE MOLECULE PROTEIN IDENTIFICATION THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2016-08-18 US claimed
WO-2015042506-A1 HIGH-THROUGHPUT SINGLE MOLECULE PROTEIN IDENTIFICATION THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-03-26 WO claimed
US-20080014595-A1 Detection of glutathionylated proteins THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2008-01-17 US claimed
WO-2007087365-A2 DETECTION OF GLUTATHIONYLATED PROTEINS UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2007-08-02 WO claimed
US-20050250170-A1 Determination of metal ions in solution by photoluminescence anisotropy THOMPSON, RICHARD B. 2005-11-10 US claimed
WO-2005101019-A2 DETECTION OF NITROSYLATED PROTEINS UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2005-10-27 WO claimed
US-20020055091-A1 Determination of metal ions in solution by photoluminescence anisotropy UNIVERSITY OF PENNSYLVANIA 2002-05-09 US claimed
EP-0914392-B1 LUMINESCING INKS AND USE OF SUCH INKS IN CODING AND OTHER MARKING OPERATIONS POST OFFICE (GB) 2000-10-25 EP claimed
EP-0715721-B1 PHOSPHATE ASSAY MEDICAL RES COUNCIL (GB) 1999-11-10 EP claimed
US-5601809-A USING A SULFHYDRYL REACTANT THE GILLETTE COMPANY (US) 1997-02-11 US claimed
EP-0715721-A1 PHOSPHATE ASSAY MEDICAL RESEARCH COUNCIL (GB) 1996-06-12 EP claimed
WO-1995002825-A1 PHOSPHATE ASSAY MEDICAL RESEARCH COUNCIL (GB) 1995-01-26 WO claimed