SCHEMBL25568634

SCHEMBL25568634

CC(C)(C)OC(=O)NC1(CCCN)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34
CTSL P07711 1/20 0.34
APLNR P35414 1/20 0.33
PPIA P62937 1/20 0.33
P2RX7 Q99572 1/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA7 P43166 1/20 0.32
CTSK P43235 1/20 0.31
DRD2 P14416 2/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
ITGB3 P05106 2/20 0.31
ITGA2B P08514 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364824 0.90 MEN1 (0.36) TDP1MAOAMAOBMEN1KMT2A
Hydrochloric Acid SCHEMBL30426524 0.89 MEN1 (0.35) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL28220352 0.88 P2RX7 (0.40) P2RX7ITGB3ITGA2BEPHX1
SCHEMBL4760970 0.85 TDP1 (0.47) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL25574885 0.84 P2RX7 (0.38) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL3365305 0.84 P2RX7 (0.40) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL24845266 0.84 TDP1 (0.50) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL1752478 0.83 MEN1 (0.37) TDP1MAOAMAOBMEN1KMT2A
Hydrochloric Acid SCHEMBL28213668 0.81 MEN1 (0.36) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL3369497 0.81 TDP1 (0.42) TDP1MEN1KMT2AGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250019376-A1 CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS MERCK SHARP & DOHME LLC (US) 2025-01-16 US disclosed
EP-4433476-A1 CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS Merck Sharp & Dohme LLC (US) 2024-09-25 EP disclosed
US-11932637-B2 Chromane amidine monobactam compounds for the treatment of bacterial infections MERCK SHARP & DOHME LLC (US) 2024-03-19 US disclosed
US-20230159517-A1 CHROMANE AMIDINE MONOBACTAM COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS MERCK SHARP & DOHME LLC (US) 2023-05-25 US disclosed
US-20230159517-A1 CHROMANE AMIDINE MONOBACTAM COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS MERCK SHARP & DOHME LLC (US) 2023-05-25 US disclosed
US-20230159517-A1 CHROMANE AMIDINE MONOBACTAM COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS MERCK SHARP & DOHME LLC (US) 2023-05-25 US disclosed
WO-2023091438-A1 CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS MERCK SHARP & DOHME LLC (US) 2023-05-25 WO disclosed
WO-2023091438-A1 CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS MERCK SHARP & DOHME LLC (US) 2023-05-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159517-A1 CHROMANE AMIDINE MONOBACTAM COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS TCOF1, SLC10A2, PAM TDP1 3270/4885MAOA 2075/4885MAOB 1629/4885
US-20250019376-A1 CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS PAM, ACMSD, MGAM2 TDP1 4222/4885MAOA 382/4885MAOB 293/4885
US-11932637-B2 Chromane amidine monobactam compounds for the treatment of bacterial infections MGAM, MGAM2, ELANE TDP1 3311/4885MAOA 995/4885MAOB 421/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.