SCHEMBL2563095

SCHEMBL2563095

COc1ccc(NC2CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
GAA P10253 4/20 0.54
MAPT P10636 4/20 0.54
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
KDM4E B2RXH2 2/20 0.54
THRB P10828 1/20 0.54
MAPK1 P28482 1/20 0.54
RECQL P46063 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
CCR6 P51684 2/20 0.51
GFER P55789 1/20 0.49
MERTK Q12866 1/20 0.49
TSHR P16473 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13450514 0.92 ALDH1A1 (0.50) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL3108892 0.92 RAB9A (0.57) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL7790492 0.91 ALDH1A1 (0.52) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL674674 0.90 RAB9A (0.59) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL3121134 0.87 ALDH1A1 (0.49) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL4140224 0.87 HTR6 (0.57) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL31152659 0.85 POLB (0.65) ALDH1A1GAAMAPTKDM4ENPSR1
SCHEMBL9822760 0.81 ALDH1A1 (0.45) ALDH1A1MAPTNPC1RAB9ATDP1
SCHEMBL24538113 0.79 ALDH1A1 (0.65) ALDH1A1MAPTNPC1RAB9AMAPK1
SCHEMBL24537639 0.79 ALDH1A1 (0.65) ALDH1A1MAPTNPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064493-A1 COMPOUNDS AND METHODS FOR TREATING CORONAVIRUSES Clear Creek Bio, Inc. (US) 2023-04-20 WO disclosed
CN-112898173-B Method for preparing amide compound by photocatalytic organic amine 湖南中医药大学 2022-10-11 CN disclosed
CN-109153636-B Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors 朱比连特埃皮科尔有限责任公司 2021-10-22 CN disclosed
CN-112898173-A Method for preparing amide compound by photocatalytic organic amine 湖南中医药大学 2021-06-04 CN disclosed
WO-2019016385-A1 BENZAMIDE COMPOUNDS AND THEIR USE AS HERBICIDES BASF SE (DE) 2019-01-24 WO disclosed
CN-109153636-A Cyclopropyl-amide compound as dual LSD1/HDAC inhibitor 朱比连特比利斯有限公司 2019-01-04 CN disclosed
US-8741934-B2 Inhibitors of ion channels PFIZER LIMITED (GB) 2014-06-03 US disclosed
CN-102863341-B Chemical synthesis method of (1R, 2S)-2-aryl cyclopropylamine derivative UNIV NANTONG 2014-05-07 CN disclosed
US-20130072471-A1 Inhibitors of Ion Channels MARRON BRIAN EDWARD (US) 2013-03-21 US disclosed
EP-2560978-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS Mars, Incorporated (US) 2013-02-27 EP disclosed
US-8357711-B2 Heterocyclic sulfonamides as inhibitors of ion channels PFIZER LIMITED (GB) 2013-01-22 US disclosed
CN-102863341-A Chemical synthesis method of (1R, 2S)-2-aryl cyclopropylamine derivative UNIV NANTONG 2013-01-09 CN disclosed
WO-2011133653-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED (US) 2011-10-27 WO disclosed
US-20090143358-A1 INHIBITORS OF ION CHANNELS ICAGEN, INC. (US) 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130072471-A1 Inhibitors of Ion Channels TRPV1, TRPV5, TRPA1 ALDH1A1 3113/4885GAA 3679/4885MAPT 2938/4885
US-20090143358-A1 INHIBITORS OF ION CHANNELS TRPV1, TRPV5, TRPA1 ALDH1A1 3113/4885GAA 3679/4885MAPT 2938/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.