SCHEMBL2564222

SCHEMBL2564222

O=C(Nc1ccncc1)c1c(Cc2ccc(F)cc2)[nH]c2ccc(Br)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.44
ALDH1A1 P00352 4/20 0.44
NPSR1 Q6W5P4 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 1/20 0.41
LMNA P02545 3/20 0.40
POLB P06746 1/20 0.40
LRRK2 Q5S007 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
NOD2 Q9HC29 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5533925 0.79 MAPT (0.46) HTTALDH1A1NPSR1SMN1; SMN2MAPK1
SCHEMBL5532547 0.76 MAPT (0.45) HTTALDH1A1TDP1SMN1; SMN2LMNA
SCHEMBL5535769 0.75 GABRP (0.42) HTTALDH1A1SMN1; SMN2MAPK1POLB
SCHEMBL8805923 0.75 ROCK2 (0.45) HTTALDH1A1NPSR1SMN1; SMN2MAPK1
SCHEMBL5526963 0.73 ALOX5 (0.42) HTTALDH1A1NPSR1SMN1; SMN2MAPK1
SCHEMBL8806089 0.71 CNR1 (0.45) ALDH1A1LMNA
SCHEMBL8805163 0.69 EGFR (0.53) HTTALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL8805594 0.69 ROCK2 (0.48) ALDH1A1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL8805331 0.69 NPY5R (0.42) ALDH1A1NPSR1SMN1; SMN2MAPK1LMNA
SCHEMBL7416262 0.68 ACHE (0.44) HTTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011133862-A1 METHODS AND COMPOSITIONS FOR PROMOTING MYELINATION OREGON HEALTH AND SCIENCE UNIVERSITY (US) 2011-10-27 WO claimed
WO-2011133862-A1 METHODS AND COMPOSITIONS FOR PROMOTING MYELINATION OREGON HEALTH AND SCIENCE UNIVERSITY (US) 2011-10-27 WO disclosed